| Cat. No. |
Product Name |
Information |
| PC-61743 |
MRS2179
P2Y1 antagonist
|
MRS2179 is a potent, selective, competitive P2Y1 receptor antagonist with Kb of 100 nM. |
| PC-61587 |
Elinogrel
P2Y12 antagonist
|
Elinogrel (PRT060128) is a selective, reversible, competitive and direct-acting P2Y12 receptor antagonist with IC50 of 20 nM. |
| PC-61586 |
BX 667
P2Y12 antagonist
|
BX 667 is a potent P2Y12 receptor antagonist that blocks ADP-induced platelet aggregation in human, dog and rat blood (IC50=97, 317 and 3000 nM respectively). |
| PC-61585 |
Cangrelor tetrasodium
P2Y12 antagonist
|
Cangrelor tetrasodium (AR-C69931MX) is a potent, selective P2T/P2Y12 receptor antagonist with IC50 of 0.4 nM against ADP-induced aggregation of human platelets. |
| PC-61584 |
Cangrelor
P2Y12 antagonist
|
Cangrelor (AR-C69931MX) is a potent, selective P2T/P2Y12 receptor antagonist with IC50 of 0.4 nM against ADP-induced aggregation of human platelets. |
| PC-61535 |
SAR216471 hydrochloride
P2Y12 antagonist
|
SAR216471 hydrochloride is a potent, highly selective, intravenous and oral, reversible P2Y12 receptor antagonist with binding IC50 of 17 nM. |
| PC-61413 |
BPTU
P2Y1 antagonist
|
BPTU (BMS-646786) is a potent, highly selective and allosteric antagonist of P2Y1 receptor with Ki of 6 nM for hP2Y1. |
| PC-61412 |
MRS2500
P2Y1 antagonist
|
MRS2500 is a highly potent and selective antagonist of the platelet P2Y1 receptor with Ki of 0.78 nM. |
| PC-61411 |
MRS2500 tetraammonium
P2Y1 antagonist
|
MRS2500 tetraammonium is a highly potent and selective antagonist of the platelet P2Y1 receptor with Ki of 0.78 nM. |
| PC-61410 |
MRS-2365
P2Y1 agonist
|
MRS-2365 is a highly potent, selective P2Y1 receptor agonist with EC50 of 1.2 nM. |
| PC-46930 |
Suramin
Cullin-RING E3 ubiquitin ligase inhibitor
|
Suramin sodium salt (BAY-205, NF-060) is an antitrypansomal drug that also possesses antitumor activity, inhibits CRL (Cullin-RING E3 ubiquitin ligases) activity by disrupting its ability to recruit Cdc34. |
| PC-45275 |
Clopidogrel hydrogen sulfate
P2Y12 antagonist
|
Clopidogrel hydrogen sulfate is a thienopyridine-class antiplatelet agent that works by irreversibly inhibiting P2Y12 receptor on platelets. |
