| Cat. No. |
Product Name |
Information |
| PC-21834 |
CD2019
RARβ agonist
|
CD2019 is a selective retinoic acid receptor β (RARβ) agonist, CD2019 is 5-fold selective for RARβ over RARα and 12-fold selective for RARβ over RARγ. |
| PC-21833 |
ER-38925
RARα agonist
|
ER-38925 is a potent, selective retinoic acid receptor subtype α (RAR-α) agonist, inhibits proliferation of mouse spleen cells with IC50 of 0.2 nM. |
| PC-21720 |
RXR agonist 33
RXR agonist
|
RXR agonist 33 is a highly potent, selective and partial RXR agonist with EC50 of 9/18/11 nM for RXRα/β/γ respectively. |
| PC-20840 |
BPA-B9
RXRα inhibitor
|
BPA-B9 (Bipyridine amide B9) is a small molecule RXRα-targeted anti-mitotic agent, binds to RXRα (Kd=39 nM) and selectively inhibits the p-RXRα/PLK1 interaction to induce mitotic arrest and catastrophe in cancer cells. |