| Cat. No. |
Product Name |
Information |
| PC-70289 |
CD 1530
RARγ agonist
|
CD 1530 is a potent and selective RARγ receptor agonist with Ki of 150 nM, >10-fold less potent for RARβ and RARα. |
| PC-70288 |
BMS-753
RARα agonist
|
BMS-753 (BMS753) is a potent, specific RARα agonist with Ki of 2 nM, displays no significant effects on RARγ in reporter based assays. |
| PC-70122 |
AGN-195183
RARα agonist
|
AGN-195183 (VTP-195183;NRX-195183, IRX-5183) is a potent, selective RARα agonist with binding Kd of 3 nM. |
| PC-42609 |
AM580
RARα agonist
|
AM580 (CD336, NSC608001, Ro 40-6055) is an analog of retinoic acid that fuctions as a selective RARα agonist with EC50 of 0.3 nM. |
| PC-42316 |
AR7
|
AR7 (AR-7, AR 7) is a novel retinoid derivative that functions as chemical activator on RARα activity. |
| PC-21837 |
E6060
RARα agonist
|
E6060 is a potent, selective retinoic acid receptor subtype α (RAR-α) agonist with Ki of 0.2 nM, IC50 of 0.2 nM for RAR-α-mediated reporter transactivation assays. |
| PC-21835 |
CD2665
RARγ inhibitor
|
CD2665 is a potent, selective and orally active RAR-β/ RAR-γ antagonist with Ki of 306 and 110 nM, respectively. |
| PC-21834 |
CD2019
RARβ agonist
|
CD2019 is a selective retinoic acid receptor β (RARβ) agonist, CD2019 is 5-fold selective for RARβ over RARα and 12-fold selective for RARβ over RARγ. |
| PC-21833 |
ER-38925
RARα agonist
|
ER-38925 is a potent, selective retinoic acid receptor subtype α (RAR-α) agonist, inhibits proliferation of mouse spleen cells with IC50 of 0.2 nM. |
| PC-21720 |
RXR agonist 33
RXR agonist
|
RXR agonist 33 is a highly potent, selective and partial RXR agonist with EC50 of 9/18/11 nM for RXRα/β/γ respectively. |
| PC-21210 |
BMS961
RARgamma agonist
|
BMS961 is a potent, selective retinoic acid receptor-gamma (RARγ) agonist. |
| PC-21164 |
IRX4647
RARγ agonist
|
IRX4647 is a selective RARγ agonist, regulates T cell biology and reduces syngeneic tumor growth of immune checkpoint-resistant lung cancer cell line (344SQ) when combined with anti-PD-L1. |
