SRPK compound (inhibitors, antagonists, modulators)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-49773	MSC-1186 SRPK inhibitor	MSC-1186 (MSC2711186) is a potent, highly selective pan-SRPK inhibitor with I50 of 2.7 nM, 81 nM and 0.6 nM against SRPK1, SRPK2 and SRPK3, respectively.
PC-49772	SRPIN340 SRPK1 inhibitor	SRPIN340 (SRPIN 340) is a potent, highly selective inhibitor of serine-arginine-rich protein kinase (SRPK1) with Ki value of 0.89 uM (SRPK1).
PC-35908	SPHINX31 SRPK1 inhibitor	SPHINX31 (SPHINX 31) is a potent, selective, ATP competitive inhibitor of Serine/arginine-protein kinase 1 (SRPK1) with IC50 of 5.9 nM.
PC-63234	SRPKIN-1 SRPK1/2 inhibitor	SRPKIN-1 (JH-XI-05-01) is a potent, selective, covalent SRPK1/2 inhibitor with IC50 of 35.6/98 nM, respectively.
PC-60568	SRPIN803 SRPK1/CK2 inhibitor	SRPIN803 is a novel small molecule dual inhibitor of SRPK1 and CK2 with IC50 of 2.4 uM and 0.2 uM, respectively, does not inhibit SRPK2.
PC-49774	SRPK1 inhibitor DBS1 SRPK1 inhibitor	SRPK1 inhibitor DBS1 (Docking Blocker of SRPK1) is a 20-mer peptide, cell-penetrating, non-ATP-competitive inhibitor of SRPK1 with ITC Kd of 5.6 uM, inhibits kinase activity of SRPK1 in a competitive manner against the substrate SRSF1 (Ki=2.12 uM), but not ATP.

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