| Cat. No. |
Product Name |
Information |
| PC-60221 |
G-9791
group I PAK inhibitor
|
G-9791 (G9791) is a potent and selective group I PAK (pan-PAK1/2/3) inhibitor with Ki of 0.95/2 nM for PAK1/2, respectively. |
| PC-45665 |
G-5555
PAK1 inhibitor
|
G-5555 is a potent and selective p21-activated kinase 1 (PAK1) inhibitor (Ki=3.7 nM). |
| PC-45644 |
FRAX-1036
PAK inhibitor
|
FRAX1036 is a potent and selective inhibitor of group I PAKs (PAK1, Ki=23.3 nM; PAK2, Ki=72.4 nM). |
| PC-46979 |
Hydrastine
PAK4 inhibitor
|
An alkaloid of Hydrastis canadensis used in many dietary supplements intended to enhance the immune system. |
| PC-44510 |
FRAX597
PAK inhibitor
|
FRAX597 is a potent, selective ATP-competitive inhibitor of group I PAKs with IC50 of 8/13/19 nM for PAK1/2/3. |
| PC-49534 |
NVS-PAK1-1
PAK1 inhibitor
|
NVS-PAK1-1 is a potent, selective and allosteric inhibitor of PAK1 with IC50 of 5 nM, potently inhibits PAK1 phosphorylation in vitro and in vivo. |
| PC-73199 |
FRAX486
group I PAKs inhibitor
|
FRAX486 is potent, selective, brain-penetrant group I PAKs inhibitor with IC50 of 8.25, 39.5, and 55.3 nM for PAK1, PAK2 and PAK3, respectively. |
