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Request The Product List ofAryl hydrocarbon Receptor (AhR) Aryl hydrocarbon Receptor (AhR)

Cat. No. Product Name Information
PC-38860

IK-175

AhR inhibitor

IK-175 is a potent, selective and orally active aryl hydrocarbon receptor (AHR) antagonist with IC50 of 91 nM in human HepG2 cells expressing an AHR-dependent DRE-luciferase reporter and stimulated with 80 nM of the AHR agonist VAF347.
PC-38065

BAY2416964

AHR antagonist

BAY2416964 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist with IC50 of 341 nM.
PC-61627

FICZ

AhR agonist

FICZ is a high affinity aryl hydrocarbon receptor (AhR) agonist with Kd of 70 pM.
PC-60777

Phortress

AhR agonist

Phortress (NSC710305) is the L-lysylamide prodrug of 5F-203 (NSC703786), a potent, selective antitumour agent through activation the aryl hydrocarbon receptor (AhR) pathway.
PC-60776

5F 203

5F 203 (NSC 703786) is a potent, selective antitumour agent through activation the aryl hydrocarbon receptor (AhR) pathway.
PC-45600

ITE

A endogenous ligand, potent aryl hydrocarbon receptor (AhR) agonist in vitro.
PC-21584

iCDM-34

AhR agonist

iCDM-34 is a small molecule inhibitor with anti-HCV and anti-HBV activities, suppresses HBV DNA and acts as an aryl hydrocarbon receptor (AhR) agonist.
PC-21481

GDU-952

AhR agonist

GDU-952 is a novel small molecule aryl hydrocarbon receptor (AhR) agonist, activates and induces nuclear translocation of AhR.
PC-38597

KYN-101

AhR antagonist

KYN-101 (KYN101) is a potent, selective synthetic antagonist of aryl hydrocarbon receptor (AHR) with IC50 of 22 nM in human HepG2 DRE-luciferase reporter assay and 23 nM in murine Hepa1 Cyp-luc assay.
PC-38513

SGA360

AhR modulator

SGA360 is a high-affinity, selective modulator of aryl hydrocarbon receptor (AhR), competitively binds to AhR (IC50 =3 uM) and represses serum amyloid A 1 (SAA1) gene expression induced by IL-1β in Huh7 cells.
PC-43148

CH-223191

CH-223191 is a potent, specific antagonist of AhR (aryl hydrocarbon receptor), potently inhibits TCDD-induced AhR-dependent transcription with IC50 of 0.03 uM.
PC-61319

TCDD

A potent AHR (aryl hydrocarbon receptor) agonist that induces degradation of AhR by the ubiquitin-proteasome pathway.

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