| Cat. No. |
Product Name |
Information |
| PC-21691 |
ART26.12
FABP5 inhibitor
|
ART26.12 is a third generation, selective fatty acid-binding protein 5 (FABP5) inhibitor with Ki value of 0.77 uM, >25-fold selective over FABP3, FABP4 and FABP7. |
| PC-61187 |
FABP4 inhibitor 1
FABP4 inhibitor
|
FABP4 inhibitor 1 is a potent, selective Fatty acid-binding protein (FABP4, aP2) inhibitor with Ki of 30 nM. |
| PC-61186 |
HTS01037
A-FABP/aP2 inhibitor
|
HTS01037 is a highly potent ligand of adipocyte fatty acid binding protein (A-FABP/aP2) with Ki of 0.67 uM. |
| PC-42435 |
BMS-309403
FABP4 inhibitor
|
BMS-309403 is a potent, selective, cell-permeable and orally active inhibitor of FABP4 (Fatty acid binding protein 4) with Ki of < 2 nM. |
| PC-25549 |
RO6806051
FABP4/5 inhibitor
|
RO6806051 is a potent, selective, dual fatty acid binding protein 4 and 5 (FABP4 and FABP5) inhibitor with Ki of 11 nM and 86 nM for hFABP4 and hFABP5 respectively, shows good selectivity over FABP3. |
| PC-25492 |
FABP inhibitor MF6
FABP5/FABP7 inhibitor
|
FABP inhibitor MF6 (FABP ligand 6) is a small molecule ligand / inhibitor of fatty acid-binding proteins (FABPs) with high affinity for FABP7 (Kd=20 nM), with much weaker affinity for FABP3 (Kd=1038 nM) and FABP5 (Kd=874 nM). |
| PC-23932 |
CRE-14
FABP4 inhibitor
|
CRE-14 is a specific, high affinity inhibitor of fatty acid-binding protein 4 (FABP4) with Kd of 654 nM in MST assays, impairs coronavirus replication. |
| PC-22077 |
FABP1 inhibitor 44
FABP1 inhibitor
|
FABP1 inhibitor 44 is a highly selective, first-in-class FABP1 inhibitor with IC50 of 4.46 uM, does not inhibit other subtypes of FABP (FABP3/4). |
| PC-38573 |
FABP4/5 inhibitor compound 3
FABP4/5 inhibitor
|
FABP4/5 inhibitor compound 3 is a potent dual FABP4 and FABP5 inhibitor with Kd of 0.02 and 0.56 uM, respectively. |
| PC-38572 |
FABP4/5 inhibitor compound 2
FABP4/5 inhibitor
|
FABP4/5 inhibitor compound 2 is a potent dual FABP4 and FABP5 inhibitor with Kd of 0.01 and 0.52 uM, respectively, reduces isoproterenol-stimulated lipolysis in mouse 3T3-L1 adipocytes with IC50 of 22 uM. |
