| Cat. No. |
Product Name |
Information |
| PC-60954 |
Eribaxaban
FXa inhibitor
|
Eribaxaban (PD-0348292) is a potent, selective and orally efficacious factor Xa (FXa) inhibitor with IC50 of 0.32 nM. |
| PC-45940 |
Otamixaban
FXa inhibitor
|
Otamixaban (FXV-673, FXV673) is potent and selective factor Xa (FXa) inhibitor with Ki of 0.4 nM. |
| PC-42504 |
Edoxaban tosylate monohydrate
FXa inhibitor
|
Edoxaban tosylate monohydrate (DU-176b) is a potent and orally active Factor Xa (FXa) inhibitor with Ki of 0.561 nM. |
| PC-42503 |
Edoxaban tosylate
FXa inhibitor
|
Edoxaban tosylate (DU-176b) is a potent and orally active Factor Xa inhibitor with Ki of 0.561 nM. |
| PC-42502 |
Edoxaban
FXa inhibitor
|
Edoxaban (DU-176) is a potent and orally active Factor Xa (FXa) inhibitor with Ki of 0.561 nM. |
| PC-45832 |
Apixaban
FXa inhibitor
|
Apixaban (BMS-562247) is a highly potent, selective, efficacious, and orally bioavailable inhibitor of factor Xa (FXa) with Ki of 0.08 nM. |
| PC-42505 |
Betrixaban
FXa inhibitor
|
Betrixaban (PRT054021) is a highly potent, selective Factor Xa (FXa) inhibitor with Ki/IC50 of 0.117 nM/1.5 nM. |
| PC-45897 |
Rivaroxaban
FXa inhibitor
|
Rivaroxaban (BAY 59-7939) is a highly potent and selective, direct FXa inhibitor with IC50 of 0.7 nM. |
| PC-24872 |
BAY-878
FIIa/Xa inhibitor
|
SATI (BAY-878) is a potent and highly selective, direct dual FIIa/Xa inhibitor with IC50 of 2.4/0.91 nM respectively. |
| PC-24866 |
Segatroxaban
FIIa/Xa inhibitor
|
Segatroxaban (SAR107375E) is a potent and highly selective dual FIIa/Xa inhibitor with Ki values of 8 nM and 1 nM on FIIa and FXa, IC50 values of 0.3/0.7 nM (FIIa/FXa) in buffer and of 16/3 nM (FIIa/FXa) in plasma, respectively. |
| PC-24865 |
RWJ-445167
FIIa/Xa inhibitor
|
RWJ-445167 (3DP-10017) is a potent, dual inhibitor of thrombin and factor Xa (FIIa/Xa inhibitor) with Ki of 4.0/230 nM respectively. |
| PC-24864 |
Tanogitran dihydrochloride
FIIa/Xa inhibitor
|
Tanogitran dihydrochloride (BIBT986) is a potent, dual inhibitor of thrombin/factor Xa with Ki values of 2.7/26 nM, respectively. |
