| Cat. No. |
Product Name |
Information |
| PC-62215 |
GSK-484 hydrochloride
PAD4 inhibitor
|
GSK-484 hydrochloride is a potent, highly selective and reversible protein arginine deiminase PAD4 inhibitor with IC50 of 80 nM in FP binding assay (0.2 mM Ca), 50 nM in PAD4 NH3 release inhibition assay. |
| PC-62214 |
GSK-484
PAD4 inhibitor
|
GSK-484 is a potent, highly selective and reversible protein arginine deiminase PAD4 inhibitor with IC50 of 80 nM in FP binding assay (0.2 mM Ca), 50 nM in PAD4 NH3 release inhibition assay. |
| PC-61919 |
Streptonigrin
PAD4 inhibitor, RAD54 inhibitor
|
Streptonigrin (Bruneomycin, NSC 45383) is a potent, selective, and irreversible PAD4 inactivator with IC50 of 1.87 uM, also binds directly to RAD54 with Kd of 9.1 uM, inhibits ATPase and DNA branch migration activity of RAD54. |
| PC-38517 |
GSK121 trifluoroacetate
PAD4 inhibitor
|
GSK121 TFA salt is a small molecule inhibitor of potein arginine deiminase 4 (PAD4) with IC50 of 3.2 uM. |
