Cat. No. |
Product Name |
Information |
PC-35836D |
d4-PGN9856
EP2 receptor agonist
|
d4-PGN9856 is a d4-labelled PGN-9856, which is a potent, selective prostaglandin EP2 receptor agonist. |
PC-20856 |
LY3127760
EP4 antagonist
|
LY3127760 is a potent, selective prostaglandin E4 (EP4) receptor antagonist with binding Ki of 58 nM (hEP4) and cAMP IC50 of 5.6 nM. |
PC-49034 |
KMN-159
EP4 agonist
|
KMN-159 is a potent, selective small-molecule full agonist of the prostaglandin E2 type 4 (EP4) receptor with Ki of 0.24 nM (rEP4) and EC50 of 10.6 nM in the BMC ALP assays, with no affinity for EP2 (Ki>10,000 nM). |
PC-38844 |
OC000459
DP2 (CRTh2) inhibitor
|
OC000459 is a potent, selective, and orally active D prostanoid receptor 2 (DP2, CRTH2) antagonist with Ki of 13/3 nM for human/recombinant DP2, respectively. |
PC-72851 |
TG8-260
EP2 antagonist
|
TG8-260 is a second-generation, potent, selective EP2 antagonist with Schild KB of 13.2 nM. |
PC-38004 |
HL-43
EP4 antagonist
|
HL-43 (EP4 antagonist HL-43) is a selective prostaglandin E receptor 4 (EP4) antagonist, promotes chondrocyte differentiation/cartilage regeneration and anabolism with low toxicity. |
PC-36058 |
BGC20-1531
EP4 antagonist
|
BGC20-1531 (PGN-1531, AP 1531) is a potent, selective prostanoid EP receptor EP antagonist, exhibits high affinity at recombinant human EP4 receptors expressed in cell lines (pKB=7.6) and native EP4 receptors in human cerebral and meningeal artery (pKB=7.6-7.8). |
PC-36057 |
BAY-1316957
|
BAY-1316957 (BAY 1316957) is a highly potent, selective, orally available human prostaglandin E2 receptor subtype 4 (hEP4-R) antagonist with IC50 of 15.3 nM. |
PC-35836 |
PGN-9856
EP2 receptor agonist
|
PGN-9856 (PGN9856) is a novel potent, selective prostaglandin EP2 receptor agonist with pKi of > 8.3, shows high selectivity over EP1 , EP3 , EP4 , DP, FP, IP and TP receptors. |
PC-35786 |
TG8-69
EP2 antagonist
|
TG8-69 is a peripherally restricted, highly potent, selective, aqueous-soluble EP2 antagonist with Kb of 48.5 nM. |
PC-35542 |
ASP7657
EP4 antagonist
|
ASP7657 (ASP-7657) is a potent, selective, orally active prostaglandin EP4 receptor antagonist with Ki values of 6.02 nM and 2.21 nM for rat and human EP4 receptors, resepctively. |
PC-35221 |
CR6086 sodium
EP4 antagonist
|
CR6086 sodium (CR-6086) is a potent, selective prostaglandin E2 receptor 4 (EP4) antagonist with Ki of 16.6 nM (hEP4 receptor), inhibits PGE2-stimulated cAMP production with IC50 of 22 nM. |