| Cat. No. |
Product Name |
Information |
| PC-42387 |
PGD2-IN-1
PGD2 antagonist
|
PGD2-IN-1 is a potent prostaglandin D2 receptor (PGD2, DP) receptor antagonist with IC50 of 0.3 nM. |
| PC-45826 |
Laropiprant
DP1 antagonist
|
Laropiprant (MK-0524) is a potent and selective prostaglandin D2 (PGD2) receptor (DP1) antagonist with Ki of 0.57 nM. |
| PC-45103 |
GW627368
EP4 antagonist
|
GW627368 is a potent and selective competitive antagonist of prostanoid EP4 receptor with pKi of 7.0. |
| PC-45111 |
TG6-10-1
EP2 antagonist
|
TG6-10-1 is a potent and selective antagonist of prostaglandin E2 receptor subtype EP2 with Kb of 17.8 nM. |
| PC-45579 |
PF-04418948
EP2 antagonist
|
PF-04418948 (PF 04418948) is a novel potent and selective prostaglandin EP2 receptor antagonist. |
| PC-45077 |
Grapiprant
EP4 antagonist
|
Grapiprant (CJ-023423, AAT-007) is a potent, selective EP4 receptor antagonist with Ki values of 13/20 nM against human and rat EP(4) receptors. |
| PC-42573 |
MK-2894 sodium
EP4 antagonist
|
MK-2894 sodium is a highly potent, selective, second generation prostaglandin E2 subtype 4 receptor (EP4) antagonist with Ki of 0.56 nM. |
| PC-42572 |
MK-2894
EP4 antagonist
|
MK-2894 (MK2894) is a highly potent, selective, second generation prostaglandin E2 subtype 4 receptor (EP4) antagonist with Ki of 0.56 nM. |
| PC-27072 |
Evatanepag
EP2 receptor agonist
|
Evatanepag (CP-533536, CP-533,536) is a highly selective and potent functional EP2 receptor agonist with high affinity to rat EP2 receptor (IC50=50 nM), is >50-fold more selective over EP4 receptor subtype. |
| PC-27006 |
TP-18
EP2/EP4 antagonist
|
TP-18 is a potent, selective, orally available dual PGE2 receptor EP2/EP4 antagonist with IC50 of 9.5/3.3 nM respectively. |
| PC-26606 |
SC-51089
EP1 antagonist
|
SC-51089 (SC51089) is a selective antagonist of prostaglandin E2 EP1 receptor, with Ki values of 1.3, 11.2, 17.5, and 61.1 μM for EP1, TP, EP3, and FP receptors, respectively, exhibits neuroprotective activity. |
| PC-26564 |
BPN-37440
EP2 antagonist
|
BPN-37440 is a potent, selective prostaglandin-E2 receptor EP2 antagonist with IC50 of 53 nM, with no activity against DP1, EP4 and IP receptors. |
