Cat. No. |
Product Name |
Information |
PC-45075 |
Fevipiprant
CRTH2 inhibitor
|
Fevipiprant (NVP-QAW039, QAW-039) is a potent, selective, slowly dissociating CRTh2 antagonist with Kd of 1.14 nM. |
PC-42700 |
CJ-042794
EP4 antagonist
|
CJ-042794 (CJ-42794) is a potent, selective prostaglandin E receptor subtype 4 (EP4) antagonist with pKi of 8.5. |
PC-42699 |
MF498
EP4 antagonist
|
MF498 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist with Ki of 0.74 nM. |
PC-46004 |
MRE-269
IP receptor inhibitor
|
MRE-269 (ACT-333679) is a potent, selective IP receptor (prostaglandin I2 receptor) agonist with Ki of 20 nM. |
PC-45896 |
ONO-AE3-208
EP4 antagonist
|
ONO-AE3-208 (AE3-208) is a potent, selective EP4 receptor antagonist with Ki of 1.3 nM. |
PC-45118 |
Terutroban
Prostanoid TP receptor antagonist
|
Terutroban (S-18886) is a potent, selective antagonist of the thromboxane receptor (Prostanoid TP receptor) that blocks thromboxane induced platelet aggregation and vasoconstriction. |
PC-42387 |
PGD2-IN-1
PGD2 antagonist
|
PGD2-IN-1 is a potent prostaglandin D2 receptor (PGD2, DP) receptor antagonist with IC50 of 0.3 nM. |
PC-45826 |
Laropiprant
DP1 antagonist
|
Laropiprant (MK-0524) is a potent and selective prostaglandin D2 (PGD2) receptor (DP1) antagonist with Ki of 0.57 nM. |
PC-45103 |
GW627368
EP4 antagonist
|
GW627368 is a potent and selective competitive antagonist of prostanoid EP4 receptor with pKi of 7.0. |
PC-45111 |
TG6-10-1
EP2 antagonist
|
TG6-10-1 is a potent and selective antagonist of prostaglandin E2 receptor subtype EP2 with Kb of 17.8 nM. |
PC-45579 |
PF-04418948
EP2 antagonist
|
PF-04418948 (PF 04418948) is a novel potent and selective prostaglandin EP2 receptor antagonist. |
PC-45077 |
Grapiprant
EP4 antagonist
|
Grapiprant (CJ-023423, AAT-007) is a potent, selective EP4 receptor antagonist with Ki values of 13/20 nM against human and rat EP(4) receptors. |