| Cat. No. |
Product Name |
Information |
| PC-42433 |
TG 100801
Src inhibitor
|
The prodrug of TG 100572, a potent, dual receptor tyrosine kinase/Src kinase inhibitor with IC50 of 2-16 nM for VEGFR, FGFR and PDGFR, 0.1-5 nM for Src family. |
| PC-42561 |
PD173955
Src inhibitor
|
PD173955 is a potent, selective, ATP-competitive Src family kinases inhibitor with IC50 of 22 nM for Src. |
| PC-42475 |
Saracatinib
Src/Abl inhibitor
|
Saracatinib (AZD0530) is a potent, highly selective, orally available, dual Src/Abl kinase inhibitor with IC50 of 2.7, 4, 4 and 30 nM for c-Src, Yes, Lck and Abl, respectively. |
| PC-42432 |
TG 100572 hydrochloride
Src inhibitor
|
TG100572 hydrochloride is a potent, dual receptor tyrosine kinase/Src kinase inhibitor with IC50 of 2-16 nM for VEGFR, FGFR and PDGFR, 0.1-5 nM for Src family. |
| PC-42431 |
TG 100572
Src inhibitor
|
TG100572 is a potent, dual receptor tyrosine kinase/Src kinase inhibitor with IC50 of 2-16 nM for VEGFR, FGFR and PDGFR, 0.1-5 nM for Src family. |
| PC-42690 |
Lck inhibitor 2
Lck inhibitor
|
Lck inhibitor 2 uis a potent tyrosine kinases inhibitor with IC50 of 13/9/3/26/2 nM for Lck/Btk/Lyn/Syk/Txk. |
| PC-43792 |
1-Naphthyl PP1
Src inhibitor
|
1-Naphthyl PP1 (1-NA-PP1) is a potent Src family kinases with IC50 of 1.0/0.6/0.6 uM for v-Sr/c-Fyn/c-Abl. |
| PC-45084 |
T338C Src-IN-1
Src T338C inhibitor
|
T338C Src-IN-1 is a potent mutant Src T338C inhibitor with IC50 of 111 nM, exhibits 10-fold selectivity over WT c-Src. |
| PC-45085 |
T338C Src-IN-2
Src T338C inhibitor
|
T338C Src-IN-2 is a potent mutant c-Src T338C kinase inhibitor with IC50 of 317 nM, also inhibits T338C/V323A and T338C/V323S with IC50 of 57 nM/19 nM. |
| PC-45449 |
AMG-47a
Lck inhibitor
|
AMG-47a is a potent Lck kinase inhibitor with IC50 of 0.2 nM, selectively reduces the levels of EGFP-KRASG12V protein but do not affect EGFP protein in cells. |
| PC-42786 |
A-770041
Lck inhibitor
|
A-770041 (A770041) is a potent and selective small-molecule inhibitor of Lck kinase with IC50 of 147 nM. |
| PC-45439 |
KX1-004
Src inhibitor
|
KX1-004 is a non-ATP competitive Src-PTK inhibitor with IC50 of 40 uM. |
