| Cat. No. |
Product Name |
Information |
| PC-20800 |
KI-MS2-008
Max homodimer stablizer
|
KI-MS2-008 is a small molecule Max binder that modulate Myc-driven transcription in cells (IC50=1.28 uM) and inhibit viable cell levels in a Myc-dependent manner. |
| PC-20799 |
NSC13728 hydrochloride
Max homodimer stablizer
|
NSC13728 hydrochloride is a specific small molecule stabilizer of the Max homodimer inhibiting Myc function, also inhibits Myc-Max heterodimerization. |
| PC-20798 |
NSC13728
Max homodimer stablizer
|
NSC13728 is a specific small molecule stabilizer of the Max homodimer inhibiting Myc function, also inhibits Myc-Max heterodimerization. |
| PC-38695 |
MYRA-B
c-MYC inhibitor
|
MYRA-B (NSC45641) is a small molecule that induces Myc-dependent apoptosis without affecting Myc transactivation or Myc/Max DNA binding. |
| PC-38694 |
MYRA-A
c-MYC inhibitor
|
MYRA-A (NSC339585) is a small molecule Myc pathway response agent (MYRA) that inhibits Myc transactivation and interferes with the DNA-binding activity of Myc family proteins, with no effect on the E-box-binding protein USF. |
| PC-38693 |
KSI-3716
c-MYC inhibitor
|
KSI-3716 is a small molecule c-MYC inhibitor that blocks c-MYC/MAX binding to target gene promoters, inhibits c-MYC mediated transcriptional activity at concentrations as low as 1 uM. |
| PC-38661 |
L755507
c-Myc-MAX inhibitor
|
L755507 is a potent, selective β3-adrenoceptor (β3-AR) agonist, exhibits robust concentration-dependent increase in cAMP accumulation in CHO-K1 cells expressing human β3-adrenoceptors (pEC50=12.3), also effectively inhibits the c-Myc-MAX heterodimerization. |
| PC-38523 |
F1021-0686
c-Myc inhibitor
|
F1021-0686 is a novel small molecule inhibitor of c-Myc, causes the functional repression of c-Myc target gene, shows appreciable anticancer activity against c-Myc expressing cell lines (HT29, IC50=1.55 uM). |
| PC-38522 |
F0909-0360
c-Myc inhibitor
|
F0909-0360 is a novel small molecule inhibitor of c-Myc, causes the functional repression of c-Myc target gene, shows appreciable anticancer activity against c-Myc expressing cell lines (HT29, IC50=0.2 uM). |
| PC-38503 |
Mycro3
Myc inhibitor
|
Mycro3 is a selective small molecule inhibitor of Myc/Max dimerization with IC50 of 40 uM with a cognate-binding site, inhibits DNA binding of c-Myc with preference over other dimeric transcription factors in vitro. |
| PC-73141 |
MYC inhibitor EN4
MYC covalent inhibitor
|
MYC inhibitor EN4 is a covalent ligand and inhibitor of MYC, targets cysteine 171 of MYC and inhibits MYC transcriptional activity (EC50=2.8 uM). |
| PC-72260 |
PKUMDL-YC-1205
c-Myc inhibitor
|
PKUMDL-YC-1205 is a specific small molecule that can specifically bind to the disordered bHLH-LZ domain of c-Myc (SPR kd=18 uM). |
