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Cat. No. Product Name Information
PC-20522

Ibipinabant

CB1 antagonist

Ibipinabant (SLV319, BMS-646256) is a potent, selective and orally active antagonist of cannabinoid CB1 receptor with Ki of 7.8 nM, >1000-fold selectivity for CB1 over CB2.
PC-20521

PF-514273

CB1 antagonist

PF-514273 (PF 514273) is a potent, selective and orally active antagonist of cannabinoid CB1 receptor with Ki of 1.0 nM, >10000-fold selectivity for CB1 over CB2.
PC-20518

JD-5006

CB1 antagonist

JD-5006 is a potent, selective and peripherally restricted cannabinoid-1 (CB1) receptor blocker with IC50 of 18 nM, does not inhibit CB2 receptor (IC50>5000 nM).
PC-20517

JD-5037

CB1 antagonist

JD-5037 is a potent, selective and peripherally restricted cannabinoid-1 (CB1) receptor blocker with IC50 of 2 nM, does not inhibit CB2 receptor (IC50>1000 nM).
PC-20082

AM251

CB1 antagonist

AM251 (AM 251) is a potent, selective CB1 receptor antagonist (inverse agonist) with IC50 of 8 nM, Ki of 7.49 nM, displays 306-fold selectivity over CB2 receptors.
PC-20078

URB447

CB1R antagonist

URB447 (URB-447) is a peripherally restricted CB(1) antagonist/CB(2) agonist with IC50 of 313 nM (rat CB1) and 41 nM (human CB2).
PC-20077

AM6545

CB1R antagonist

AM6545 (AM-6545) is a potent, selective, oral bioavailable and non-brain-penetrant neutral CB1R antagonist with Ki of 3.3 nM, >100-fold selectivity over CB2R.
PC-20051

MRL-650

CB1R inhibitor

MRL-650 (MRL650) is a potent, selective inverse agonist of CB1 cannabinoid receptor with IC50 of <10 nM.
PC-38638

JM-00266

CB1R blocker

JM-00266 is a novel non-brain penetrant cannabinoid receptor 1 (CB1R) inverse agonist.
PC-73457

Zevaquenabant

CB1R/iNOS inhibitor

Zevaquenabant ((S)-MRI-1867) is a peripherally restricted, orally bioavailable dual CB1 receptor/iNOS inhibitor.
PC-35625

XL-001

XL-001 (XL001) is a novel specific CB2 inverse agonist with Ki of 0.5 nM.
PC-35592

AM9405

AM9405 (AM-9405, GAT-379) is novel potent, peripherally active cannabinoid type 1 (CB1) and 5-HT3 receptor agonist, inhibits the EFS-induced twitch contraction of the ileum and the colon with IC50 of 0.076 and 45.71 nM, respectively.

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