| Cat. No. |
Product Name |
Information |
| PC-43210 |
DBPR211
CB1 antagonist
|
DBPR211 (BPRCB1184, CB1-IN-4) is a potent, selective, peripherally restricted cannabinoid-1 (CB1) receptor antagonist with Ki of 0.3 nM, EC50 of 3.0 nM. |
| PC-43187 |
A-836339
CB2 agonist
|
A-836339 (A836339) is a potent and selective cannabinoid CB2 receptor agonist with Ki of 0.64 and 0.76 nM for human and rat CB2 receptors, displays 425- and 189-fold selectivity over CB1 receptor, respectively. |
| PC-63019 |
LDK1229
CB1 inverse agonist
|
LDK1229 is a novel potent, selective cannabinoid CB1 receptor inverse agonist with Ki of 220 nM. |
| PC-62915 |
MK-9470
CB1 inverse agonist
|
MK-9470 is a potent, selective cannabinoid CB1 receptor (CB1R) inverse agonist with IC50 of 0.7 nM, 18F MK-9470 has been developed for use in human brain imaging.. |
| PC-60810 |
SMM-295
CB2 agonist
|
SMM-295 is a potent, selective cannabinoid receptor 2 (CB2) agonist with Ki of 12 nM, >30-fold selectivity over CB1. |
| PC-60764 |
A 834735
Cannabinoid receptor agonist
|
A 834735 is a potent, nonselective, brain penetrant, full agonist at both the central CB1 and peripheral CB2 receptors with Ki of 4.6 and 0.31 nM, respectively. |
| PC-60763 |
JTE907
CB2 inverse agonist
|
JTE907 (JTE-907) is a potent, selective, orally active cannabinoid CB2 receptor inverse agonist with Ki of 35.9, 1.55 and 0.38 nM for human, mouse and rat CB2, respectively. |
| PC-60762 |
UR-144
CB2 agonist
|
UR-144 is a potent, selective full agonist of the peripheral cannabinoid receptor CB2 with Ki of 1.8 nM, >80-fold selectivity over CB1 (Ki=150 nM). |
| PC-60761 |
AM-2201
Cannabinoid receptor agonist
|
AM-2201 is a synthetic cannabinoid that acts as a potent, nonselective full agonist for the cannabinoid receptor with EC50 of 38 and 58 nM for CB1 and CB2, respectively. |
| PC-60760 |
AM630
CB2 antagonist
|
AM630 (6-Iodopravodoline) is a potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1. |
| PC-60759 |
AM-1221
CB1 agonist
|
AM-1221 is a potent and selective agonist for the cannabinoid receptor CB1 with Ki of 0.28 nM, 180-fold selectivity over CB2. |
| PC-60758 |
MN-25
CB2 agonist
|
CB2 agonist MN25 (AR12) is a potent, reasonably selective agonist of peripheral cannabinoid receptor with Ki of 11 nM for CB2, 22-fold selectivity over the psychoactive CB1 receptors (Ki=245 nM). |
