| Cat. No. |
Product Name |
Information |
| PC-60146 |
Olorinab
CB2 agonist
|
Olorinab (APD371) is a potent, selective and orally available CB2 cannabinoid receptor agonist with EC50 of 6.2 nM. |
| PC-60086 |
AM-6538
CB1 antagonist
|
AM-6538 (AM6538) is a potent, selective cannabinoid receptor CB1 antagonist with Ki of 5.1 nM.. |
| PC-45531 |
JD-5037
CB1 antagonist
|
JD-5037 is a potent, selective and peripherally restricted cannabinoid-1 (CB1) receptor blocker with IC50 of 2 nM, does not inhibit CB2 receptor (IC50>1000 nM). |
| PC-42171 |
Bay 59-3074
CB1/CB2 agonist
|
Bay 59-3074 is a potent, selective cannabinoid CB1/CB2 receptor partial agonist with Ki of 48.3, and 45.5 nM for human CB1 and human CB2 receptors, respectively. |
| PC-42063 |
Taranabant
CB1 inverse agonist
|
Taranabant (MK-0364) is a potent, selective and orally active cannabinoid-1 receptor (CB1R) inverse agonist with IC50 of 2.8 nM, Ki of 0.13 nM. |
| PC-42724 |
Otenabant hydrochloride
CB1 antagonist
|
Otenabant hydrochloride (CP-945598) is a potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively. |
| PC-42723 |
Otenabant
CB1 antagonist
|
Otenabant (CP-945598) is a potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively. |
| PC-42066 |
Taranabant (1R,2R) stereoisomer
|
Taranabant (1R,2R) stereoisomer is the diastereomer form of Taranabant, which is a potent, selective and orally active cannabinoid-1 receptor (CB1R) inverse agonist. |
| PC-28693 |
TXX-522
CB1R antagonist
|
TXX-522 is a potent, selective and peripherally restricted cannabinoid 1 receptor (CB1R) antagonist/inverse agonist with Ki and IC50 of 0.15 uM and 0.17 uM respectively, >100-fold selecive over CB2 receptor. |
| PC-28686 |
Surinabant
CB1R antagonist
|
Surinabant (SR147778) is a potent, selective antagonist of CB1 cannabinoid receptor (CB1R) with Ki of 0.56 nM and 3.5 nM for both the rat brain and human CB1 recombinant receptors, respectively. |
| PC-28685 |
ISAM-MM101
CB1R antagonist
|
ISAM-MM101 (CB1R antagonist 24a) is a potent, selective and peripherally directed CB1 receptor (CB1R) antagonist with Ki of 115 nM, shows high CB1R/CB2R selectivity. |
| PC-28237 |
JWH-015
CB2 agonist
|
JWH-015 is a potent, selective cannabinoid receptor 2 (CB2) agonist. |
