| Cat. No. |
Product Name |
Information |
| PC-22233 |
HU-910
CB2 agonist
|
HU-910 is a potent, selective cannabinoid CB2 receptor agonist with Ki of 6 nM in competition binding assay, IC50 of 162 nM in cAMP assay. |
| PC-22211 |
SCH225336
CB2 inverse agonist
|
SCH225336 (SCH336) is a potent, selective cannabinoid receptor CB2 inverse agonist with Ki of 0.4 nM, >2000-fold selective over CB1 receptor. |
| PC-22167 |
AM10257
CB2 antagonist
|
AM10257 is a potent, selective cannabinoid receptor 2 (CB2) antagonist with IC50 of 47 nM. |
| PC-22115 |
SMM-189
CB2 inverse agonist
|
SMM-189 is a selective cannabinoid receptor 2 (CB2) inverse agonist with Ki of 121.3 nM, 40-fold selective over CB1 receptor. |
| PC-21983 |
BAY38-7271
CB1/CB2 agonist
|
BAY 38-7271 is selective, highly potent and cannabinoid CB1/CB2 receptor agonist with 0.46-1.85 nM for rat brain, human cortex, or recombinant human CB1 receptors. |
| PC-21521 |
AM4113
CB1 neutral antagonist
|
AM4113 is a high affinity, selective cannabinoid CB1 neutral antagonist with Ki of 0.89 nM, exhibits 100-fold selectivity over CB2 receptors. |
| PC-21437 |
JWH133
CB2 agonist
|
JWH133 (JWH-133) is a potent and selective CB2 agonist with Ki of 3.4 nM, 200-fold selective over CB1 receptors, inhibits glioma growth in vivo. |
| PC-20747 |
LEI-101
CB2R agonist
|
LEI-101 (LEI 101) is a potent, selective, orally available and peripherally restricted cannabinoid CB2 receptor agonist with binding pKi of 7.5 (hCB2R). |
| PC-20521 |
PF-514273
CB1 antagonist
|
PF-514273 (PF 514273) is a potent, selective and orally active antagonist of cannabinoid CB1 receptor with Ki of 1.0 nM, >10000-fold selectivity for CB1 over CB2. |
| PC-20518 |
JD-5006
CB1 antagonist
|
JD-5006 is a potent, selective and peripherally restricted cannabinoid-1 (CB1) receptor blocker with IC50 of 18 nM, does not inhibit CB2 receptor (IC50>5000 nM). |
| PC-61396 |
Revosimeline
|
A novel potent cannabinoid receptor agonist.. |
| PC-42724 |
Otenabant hydrochloride
|
A potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively. |
