| Cat. No. |
Product Name |
Information |
| PC-60577 |
CK2 inhibitor D11
CK2α inhibitor
|
CK2 inhibitor D11 is a potent, selective, cell permeab anti-apoptotic protein kinase CK2 with Ki of 5 nM. |
| PC-60387 |
SSTC3
CK1α activator
|
SSTC3 is a novel small-molecule CK1α activator with EC50 of 30 nM (WNT-driven reporter gene assay), Kd of 32 nM. |
| PC-60386 |
VU-WS211
|
A negative control of VU-WS113, which is a potent inhibitor of Wnt signaling with EC50 of 80 nM that selectively potentiates CK1α kinase activity.. |
| PC-60385 |
VU-WS113
CK1α inhibitor
|
VU-WS113 is a potent inhibitor of Wnt signaling with EC50 of 80 nM that selectively potentiates CK1α kinase activity. |
| PC-60383 |
Pyrvinium
CK1α activator
|
Pyrvinium is an anthelmintic effective agent for pinworms that shows to be a potent inhibitor of Wnt signaling with EC50 of 10 nM, binds to all CK1 family members in vitro at low nanomolar concentrations and selectively potentiates CK1α kinase activity. |
| PC-46115 |
Pyrvinium pamoate
CK1α activator
|
Pyrvinium pamoate is an anthelmintic effective agent for pinworms that shows to be a potent inhibitor of Wnt signaling with EC50 of 10 nM, binds to all CK1 family members in vitro at low nanomolar concentrations and selectively potentiates CK1α kinase activity. |
| PC-45871 |
CX-4945 sodium salt
CK2 inhibitor
|
CX-4945 sodium salt (Silmitasertib) is a potent, selective, orally bioavailable, ATP-competitive inhibitor of protein kinase CK2 with Ki of 0.38 nM, CK2α IC50 of 1 nM. |
| PC-45870 |
CX-4945
CK2 inhibitor
|
CX-4945 (Silmitasertib, CX4945) is a potent, selective, orally bioavailable, ATP-competitive inhibitor of protein kinase Casein Kinase 2 (CK2) with Ki of 0.38 nM, CK2α IC50 of 1 nM. |
| PC-42523 |
D4476
CK1 inhibitor
|
D4476 (Casein Kinase I Inhibitor, D 4476, D-4476) is a potent, selective ATP-competitive inhibitor of CK1 with IC50 of 0.3 uM in vitro. |
| PC-42026 |
SR-3029
CK1δ/ε inhibitor
|
SR-3029 is a potent, highly selective, ATP-competitive and brain penetrating Casein Kinase 1δ/ε (CK1δ/ε) inhibitor with IC50 of 44/260 nM, respectively. |
| PC-42058 |
TA-01
CK1δ/ε inhibitor, p38α inhibitor
|
TA-01 is a potent inhibitor of Casein Kinase CK1ε, CK1δ and p38α with IC50 of 6.4, 6.8 and 6.7 nM, respectively. |
| PC-22407 |
SGC-CK2-2
CK2 inhibitor
|
SGC-CK2-2 is a potent, selective casein kinase 2 (CSNK2, CK2) chemical probe inhibitor with IC50 of 0.2 uM, shows much improved kinase selectivity compared with silmitasertib (CX-4945). |
