| Cat. No. |
Product Name |
Information |
| PC-42523 |
D4476
CK1 inhibitor
|
D4476 (Casein Kinase I Inhibitor, D 4476, D-4476) is a potent, selective ATP-competitive inhibitor of CK1 with IC50 of 0.3 uM in vitro. |
| PC-42026 |
SR-3029
CK1δ/ε inhibitor
|
SR-3029 is a potent, highly selective, ATP-competitive and brain penetrating Casein Kinase 1δ/ε (CK1δ/ε) inhibitor with IC50 of 44/260 nM, respectively. |
| PC-42058 |
TA-01
CK1δ/ε inhibitor, p38α inhibitor
|
TA-01 is a potent inhibitor of Casein Kinase CK1ε, CK1δ and p38α with IC50 of 6.4, 6.8 and 6.7 nM, respectively. |
| PC-24840 |
KDX1381
CK2α inhibitor
|
KDX1381 is a potent, selective bivalent CK2α inhibitor with IC50 of 17 nM, selecitve over a panel of over 400 protein and lipid kinases. |
| PC-24756 |
CK2 bivalent inhibitor Biv5
CK2 inhibitor
|
CK2 bivalent inhibitor Biv5 is a picomolar bivalent inhibitor of protein casein kinase 2 (CK2) with IC50 of 51 pM (CK2α), shows potent antiviral activity against SARS-CoV-2 in HEK-ACE2-TMPRSS2 and Vero cells. |
| PC-24728 |
PF-4800567
CK1ε inhibitor
|
PF-4800567 is a potent, selective inhibitor of casein kinase 1 epsilon (CK1epsilon, CK1ε) with IC50 of 32 nM, >20-fold selectivity over CK1δ. |
| PC-24636 |
Chrysoeriol
CK2 inhibitor
|
Chrysoeriol is a natural product for CK2 (Casein kinase 2) inhibitor with IC50 of 0.5 uM, inhibits JAK2/STAT3, IκB/p65, and NF-κB pathways, shows strong anti-inflammatory activities. |
| PC-24635 |
FNH79
CK2 inhibitor
|
FNH79 is a highly selective and potent CK2 (Casein kinase 2) inhibitor with IC50 of 4 nM. |
| PC-24634 |
CK2A2 inhibitor 65
CK2A2 inhibitor
|
CK2A2 inhibitor 65 is a selective, brain-penetrant inhibitor of CK2A2 and CK2A2 with IC50 of 3 nM and 4 nM respectively. |
| PC-23901 |
PF670462 dihydrochloride
CK1ε/CK1δ inhibitor
|
PF-670462 dihydrochloride (PF670462) is a potent and selective inhibitor casein kinase CK1ε and CK1δ with IC50 of 7.7 nM and 14 nM, respectively. |
| PC-23900 |
MU1742
CK1 inhibitor
|
MU1742 is a potent, selective inhibitor of Casein kinases 1 (CK1) with IC50 of 7/6/28 nM for CK1α/CK1δ/CK1ε respectively, does not inhibit p38α. |
| PC-23588 |
Fam20C inhibitor 5k
Fam20C inhibitor
|
Fam20C inhibitor 5k is a potent small-molecule Fam20C inhibitor with IC50 of 2.1 uM, showspotent anti-proliferative activity against MDA-MB-231 and BT-549 cells with IC50 values of 11.8 uM and 9.7 uM, respectively. |
