Cat. No. |
Product Name |
Information |
PC-21547 |
CKR-49-17
CK1γ2 activator
|
CKR-49-17 is a potent, allosteric small molecule activator of CK1γ2 with Kd value of 180 nM in MST assays. |
PC-20908 |
SGC-CK2-1 analog 2h
CK2α inhibitor
|
SGC-CK2-1 analog 2h is potent, selective and in vivo active inhibitor of casein kinase 2α (CSNK2A, CK2α) with pIC50 of 7.5 and 7.7 against CSNK2A1 and CSNK2A2, respectively. |
PC-20823 |
SR-4133
CK1ε inhibitor
|
SR-4133 (SR4133) is a potent and highly selective CK1ε isoform inhibitor with IC50 of 58 nM, no significant acitivity agianst CK1δ (IC50>10,000 nM). |
PC-35615 |
BMS-211
|
BMS-211 is a prodrug of the parent pan-CK2 inhibitor BMS-699.. |
PC-60384 |
Pyrvinium Iodide
|
An anthelmintic effective for pinworms that shows to be a potent inhibitor of Wnt signaling with EC50 of 10 nM, binds to all CK1 family members in vitro at low nanomolar concentrations and selectively potentiates CK1α kinase activity. |