| Cat. No. |
Product Name |
Information |
| PC-20926 |
JNJ 10191584
Histamine H4 antagonist
|
JNJ 10191584 (VUF6002) is a potent, highly selective, orally active histamine H(4) receptor antagonist with binding Ki of 26 nM, 540-fold selectivity to H4 receptor over H3 receptor. |
| PC-20925 |
JNJ 10191584 maleate
Histamine H4 antagonist
|
JNJ-10191584 (VUF6002) maleate is a potent, highly selective, orally active histamine H(4) receptor antagonist with binding Ki of 26 nM, 540-fold selectivity to H4 receptor over H3 receptor. |
| PC-49738 |
UR-MB-69
H2 receptor agonist
|
UR-MB-69 is a potent agonist of histamine H2 receptor (H2R) dopamine receptor D3R with pKi of 8.69 and 8.06, respectively. |
| PC-49737 |
UR-MB-158
H2 receptor agonist
|
UR-MB-158 is a a potent, selective H2 receptor agonist. |
| PC-49736 |
UR-Po563
H2 receptor agonist
|
UR-Po563 is a potent, selective H2 receptor agonist with pKi of 7.75, >400-fold selectivity over H1R/H3R/H4R. |
| PC-47094 |
RGH-235
H3R antagonist
|
RGH-235 is a potent, selective, and orally active H3 receptor antagonist/inverse agonist with high affinity (Ki=3.0-9.2 nM, depending on species), without affinity to H1, H2 or H4 receptors. |
| PC-72278 |
TASP0410461
H3R antagonist
|
TASP0410461 is a potent, selective histamine H3 receptor antagonist/inverse agonist. |
| PC-72277 |
Enerisant hydrochloride
H3R antagonist
|
Enerisant hydrochloride (TS091 hydrochloride) is a potent, selective histamine H3 receptor antagonist/inverse agonist with IC50 of 2.89 and 14.5 nM against hH3R and rH3R, respectively. |
| PC-72276 |
Enerisant
H3R antagonist
|
Enerisant (S091,TS-091) is a potent, selective histamine H3 receptor antagonist/inverse agonist with IC50 of 2.89 and 14.5 nM against hH3R and rH3R, respectively. |
| PC-36072 |
VUF15000
Histamine H3 agonist
|
VUF15000 (VUF-15000) is the first photoswitchable GPCR Histamine H3 receptor agonist (pKi=8.42), displays >300-fold selective for hH3R over hH1R and hH2R. |
| PC-36071 |
NLX-204
5-HT1A agonist
|
NLX-204 (NLX204) is a potent, selective, ERK1/2 phosphorylation-preferring serotonin 5-HT1A receptor agonist with pEC50 of 9.37. |
| PC-36027 |
K-8986 maleate
Histamine H1 antagonist
|
K-8986 maleate (K8986) is a histamine H1-receptor antagonist with potential therapeutic for treatment of allergic conjunctivitis. |
