| Cat. No. |
Product Name |
Information |
| PC-42514 |
GSK923295
CENP-E inhibitor
|
GSK-923295 (GSK923295) is the first potent, allosteric inhibitor of CENP-E kinesin motor ATPase activity with Ki of 3.2 nM. |
| PC-45640 |
PF-2771
CENP-E inhibitor
|
PF-2771 is a potent, selective centromere protein E (CENP-E) inhibitor with IC50 of 16.1 nM. |
| PC-45755 |
Dimethylenastron
Eg5 inhibitor
|
Dimethylenastron is a small molecule inhibitor of the mitotic kinesin Eg5. |
| PC-42308 |
Monastrol
Eg5 inhibitor
|
Monastrol is a potent, specific, allosteric and reversible mitotic kinesin Eg5 inhibitor with IC50 of 14 uM (microtubule motility inhibition). |
| PC-45861 |
Ispinesib
Eg5 inhibitor
|
Ispinesib (SB-715992) is a potent, selective, cell-permeable, allosteric inhibitor of Eg5 (mitotic kinesin KSP) with Ki of 2.3 nM. |
| PC-45767 |
K858
Kinesin Eg5 inhibitor
|
K858 is a potent, selective inhibitor of mitotic kinesin Eg5 ATPase activity with IC50 of 1.3 uM. |
| PC-22648 |
Paprotrain
KIF20A inhibitor
|
Paprotrain is a selective, reversible inhibitor of KIF20A (mitotic kinesin-like protein 2, MKLP-2, MKlp2) with Ki of 3.4 uM, does not inhibit other members of the kinesin superfamily. |
| PC-22245 |
KIF18A inhibitor compound 3
Kif18A inhibitor
|
KIF18A inhibitor compound 3 is a potent, selective mitotic kinesin KIF18A inhibitor of IC50 of 8.2 nM, inhibits KIF18A's microtubule-stimulated ATPase activity. |
| PC-21659 |
AM-1882
Kif18A inhibitor
|
AM-1882 (AM1882) is a potent, selective mitotic kinesin KIF18A inhibitor with IC50 of 230 nM in kinesin-8 microtubule (MT)-ATPase motor assays. |
| PC-21658 |
AM-9022
Kif18A inhibitor
|
AM-9022 (AM9022) is a potent, selective and orally active mitotic kinesin KIF18A inhibitor with IC50 of 47 nM in kinesin-8 microtubule (MT)-ATPase motor assays. |
