| Cat. No. |
Product Name |
Information |
| PC-70015 |
JNJ-10397049
|
A potent, selective, and bioavailable OX2 receptor antagonist with Kb of 4.5 nM. |
| PC-45062 |
Lemborexant
|
An orally active, potent, selective, dual Orexin receptor OX1/2 antagonist with binding Ki of 6/3 nM, respectively. |
| PC-45972 |
SB-408124 hydrochloride
|
A potent, selective OX1 receptor antagonist with Ki of 57 nM (whole cell assay), and 27 nM (cell membrane-based SPA assay). |
| PC-45951 |
SB-408124
|
A potent, selective OX1 receptor antagonist with Ki of 57 nM (whole cell assay), and 27 nM (cell membrane-based SPA assay). |
| PC-42159 |
TCS-OX2-29
|
A potent, selective orexin-2 receptor (OX2R) antagonist with IC50 of 40 nM. |
| PC-42732 |
SB-674042
|
A potent, selective nonpeptide Orexin 1 receptor antagonist with Ki of 26.9 nM in the membrane SPA format, and Ki of 57 nM in the whole-cell assay. |
| PC-45603 |
OX2R-Agonist-26
|
A potent, selective and non-peptide orexin receptor 2 (OX2R) agonist with EC50 of 23 nM. |
| PC-42705 |
Almorexant hydrochloride
|
A dual Orexin receptor OX1/OX2 antagonist with Ki of 1.3/0.17 nM for hOX1/hOX2 respectively. |
| PC-42704 |
Almorexant
|
A dual Orexin receptor OX1/OX2 antagonist with Ki of 1.3/0.17 nM for hOX1/hOX2 respectively. |
