TGF beta Receptor (TGFBR) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofTGF beta Receptor (TGFBR) TGF beta Receptor (TGFBR)

Cat. No.	Product Name	Information
PC-24919	LY-364947 TGFβR1 inhibitor	LY-364947 (HTS466284) is a potent ATP-competitive inhibitor of type I TGF-beta receptor kinase (TGFβR-I, ALK5) with IC50 of 59 nM, 7-fold selectivity over TGFβR-II.
PC-23416	CDD-2789 ALK2/ALK1 inhibitor	CDD-2789 is a highly potent and selective ALK2 (ACVR1)/ALK1 (ACVRL1) kinases inhibitor with Kd of 2.1/3.9 nM.
PC-22017	M4K2149 ALK2 inhibitor	M4K2149 is a potent, selective BMP type I receptor ALK2 inhibitor with IC50 of 17 nM, 34-fold selective over ALK5 (IC50=756 nM).
PC-22016	M4K2306 ALK2 inhibitor	M4K2306 is a potent, selective BMP type I receptor ALK2 inhibitor with IC50 of 7 nM, >500-fold selective over ALK5.
PC-21885	SRI-35241 TGF-β inhibitor	SRI-35241 is a potent inhibitor of thrombospondin 1 activation of TGF-β, specifically inhibits TGF-β activation mediated through TSP-1 with pIC50 of 8.12 nM, 79% inhibition at 100 nM.
PC-21884	SRI-31277 TGF-β inhibitor	SRI-31277 is a tripeptide inhibitor of thrombospondin 1 activation of TGF-β, specifically inhibits TGF-β activation mediated through TSP-1 with pIC50 of 8.28 nM.
PC-49752	Ki26894 TβR-I kinase inhibitor	Ki26894 (Ki 26894) is a small molecule TGF-beta type I receptor (TbetaR-I) kinase inhibitor, inhibits TGF-β-induced transcriptional activation in MDA-231-D-TβFluc/Rluc cells with IC50 of 0.49 uM.

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