| Cat. No. |
Product Name |
Information |
| PC-21488 |
NGD-94-1
D4R inhibitor
|
NGD-94-1 is a highly potent, selective dopamine D4 receptor antagonist with Ki of 3.6 nM. |
| PC-21487 |
Nemonapride
D2R antagonist
|
Nemonapride (YM-09151-2) is a highly potent, selective dopamine D2 receptor antagonist with Ki of 0.06 nM. |
| PC-21106 |
L-745870
D4R inhibitor
|
L-745870 (L-745,870) is is a potent, selective, brain-penetrant and orally active dopamine D4 receptor (D4R) antagonist with Ki of 0.43 nM. |
| PC-21105 |
CAB-01-019
D4R inhibitor
|
CAB-01-019 is potent, selective dopamine D4 receptor (D4R) full antagonist with binding Ki of 2.2 nM, >500-fold selectivity over D2R and D3R. |
| PC-20978 |
ZINC621433144
D4 agonist
|
ZINC621433144 is a Gi-biased, high-affinity full agonist of dopamine D4 receptor with Ki of 4.3 nM and cAMP EC50 of 0.18 nM. |
| PC-20865 |
GR-103691
D3 receptor antagonist
|
GR-103691 is a potent, selective dopamine D3 receptor antagonist with binding Ki of 0.4 nM, >100-fold selectivity over D1 and D4 receptors. |
| PC-20864 |
CJB 090
D3 receptor agonist
|
CJB 090 (CJB090) is a selective partial agonist of dopamine D3 receptor with binding Ki of 0.6 nM, CJB 090 is 97-fold selective for D3 receptors over D2. |
| PC-20863 |
NGB-2904
D3 receptor antagonist
|
NGB-2904 is a potent, highly selective dopamine D3 receptor antagonist with Ki of 2.0 nM for hD3, 56-fold selectivity over hD2. |
| PC-43162 |
Apomorphine hydrochloride hemihydrate
|
Apomorphine hydrochloride hemihydrate is a non-selective dopamine agonist which activates both D1-likeand D2-like receptors, with some preference for the latter subtypes.. |
| PC-43088 |
SKF 38393 hydrochloride
|
SKF 38393 is a potent, selective prototypical D1-like dopamine receptor with Ki of 1 and 0.5 nM for D1 and D5 receptors, shows little to no affinity for D2, D3 and D4 receptors. |
| PC-63114 |
SKF-38393 hydrobromide
|
SKF-38393 is a potent, selective D1/D5 receptor partial agonist with Ki of 1 and 0.5 nM, respectively. |
| PC-63037 |
Bromocriptine
|
Bromocriptine (2-Bromoergocriptine. |
