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Cat. No. Product Name Information
PC-23118

FOB02-04A

D3R agonist

FOB02-04A is a selective, bitopic and full agonist of dopamine 3 receptor (D3R) with Ki of 1.85 nM, 47- and 155-fold selective over D2R and D4R.
PC-23109

D5R agonist 5j

D5R agonist

D5R agonist 5j is a selective dopamine D5 receptor (D5R) partial agonist with EC50 of 269.7 nM, not active at the other four dopamine receptors.
PC-23108

PW0464

D1R agonist

PW0464 ((Rac)-Razpipadon) is a potent, selective G protein biased ligand/agonist of dopamine 1 receptor (D1R) with EC50 of 5.8 nM (Gs-cAMP), Emax of 104%.
PC-23107

PF-2562

D1R agonist

PF-2562 is a potent, selective non-catechol dopamine D1R agonist with Ki of 113 nM and EC50 of 568 nM.
PC-22633

FOB02-04

D3R agonist

FOB02-04 is a potent, selective dopamine D3 receptor (D3R) agonist with Ki of 2.84 nM, weak affinity with Ki of 106 nM for D2R.
PC-22235

Raclopride

Dopamine D2/D3 antagonist

Raclopride (FLA 870) is a potent, selective dopamine D2/D3 receptor antagonist, binds to D2 and D3 receptors with Ki of 1.8 nM and 3.5 nM, respectively.
PC-22227

A-77636 hydrochloride

Dopamine D1 agonist

A-77636 hydrochloride is a potent, selective, orally active and long acting dopamine D1 receptor agonist with Ki of 39.8 nM.
PC-22147

SCH23390 hydrochloride

Dopamine Receptor antagonist

SCH23390 hydrochloride is a potent and selective dopamine D1-like receptor antagonist with Kis of 0.2 nM and 0.3 nM for the D1 and D5 receptor, respectively.
PC-21488

NGD-94-1

D4R inhibitor

NGD-94-1 is a highly potent, selective dopamine D4 receptor antagonist with Ki of 3.6 nM.
PC-21487

Nemonapride

D2R antagonist

Nemonapride (YM-09151-2) is a highly potent, selective dopamine D2 receptor antagonist with Ki of 0.06 nM.
PC-21106

L-745870

D4R inhibitor

L-745870 (L-745,870) is is a potent, selective, brain-penetrant and orally active dopamine D4 receptor (D4R) antagonist with Ki of 0.43 nM.
PC-21105

CAB-01-019

D4R inhibitor

CAB-01-019 is potent, selective dopamine D4 receptor (D4R) full antagonist with binding Ki of 2.2 nM, >500-fold selectivity over D2R and D3R.

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