| Cat. No. |
Product Name |
Information |
| PC-61748 |
Alizapride
D2R antagonist
|
Alizapride (MS 5080) is a dopamine D2 antagonist with prokinetic and antiemetic effects used in the treatment of nausea and vomiting. |
| PC-61736 |
BP 897
D3R agonist
|
BP 897 is the first, potent, selective partial dopamine D3 receptor agonist with Ki of 0.92 nM. |
| PC-61553 |
JNJ-37822681
D2R antagonist
|
JNJ-37822681 is a potent, specific and fast-dissociating dopamine D2 antagonist with Ki of 158 nM. |
| PC-61108 |
PF-4363467
|
PF-4363467 (PF 04363467) is a novel highly potent, brain penetrant dopamine D3/D2 receptor antagonist with Ki of 1.3/692 nM respectively, with high selectivity for D3R versus other biogenic amine receptors. |
| PC-60744 |
GSK598809 hydrochloride
|
GSK598809 hydrochloride is a potent, selective, CNS penetrant and orally bioavailable dopamine D3 receptor antagonist with pKi of 8.9. |
| PC-60743 |
GSK598809
|
GSK598809 (GSK-598809) is a potent, selective, CNS penetrant and orally bioavailable dopamine D3 receptor antagonist with pKi of 8.9. |
| PC-60735 |
DETQ
Dopamine D1 modulator
|
DETQ is a novel potent, selective, allosteric and orally active dopamine D1 receptor potentiator with Kb of 26 nM. |
| PC-60665 |
SKF 83566 hydrobromide
Dopamine D1 inhibitor
|
SKF 83566 hydrobromide is a potent, selective dopamine D1 receptor antagonist with Ki of 0.56 nM. |
| PC-60614 |
A-412997 dihydrochloride
D4R agonist
|
A-412997 is a potent, selective dopamine D4 receptor agonist with Ki of 12.1 and 7.9 nM for rat and human D4 receptors, respectively. |
| PC-60216 |
PF-592379
D3R agonist
|
PF-592379 is a potent, selective, orally active agonist of dopamine D3 receptor with EC50 of 21 nM. |
| PC-70062 |
ABT-724 trihydrochloride
Dopamine D4 agonist
|
ABT-724 trihydrochloride is a potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors. |
| PC-70061 |
ABT-724
Dopamine D4 agonist
|
ABT-724 is a potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors. |
