Cat. No. |
Product Name |
Information |
PC-60614 |
A-412997 dihydrochloride
D4R agonist
|
A-412997 is a potent, selective dopamine D4 receptor agonist with Ki of 12.1 and 7.9 nM for rat and human D4 receptors, respectively. |
PC-70062 |
ABT-724 trihydrochloride
Dopamine D4 agonist
|
ABT-724 trihydrochloride is a potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors. |
PC-70061 |
ABT-724
Dopamine D4 agonist
|
A potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors. |
PC-70058 |
PD128907 hydrochloride
D3R agonist
|
PD128907 hydrochloride is a potent, selective and orally active agonist of dopamine D3 receptor (D3R) with Ki of 20 nM. |
PC-70057 |
PF-219061
|
PF-219061 (PF 219061, PF219061) is a potent, selective agonist of dopamine D3 receptor with EC50 of 8 nM. |
PC-42584 |
SKF-82958 hydrobromide
Dopamine D1 agonist, ERα agonist
|
SKF-82958 hydrobromide is a potent, full dopamine D1 agonist, produces characteristic anorectic effects, hyperactivity and self-administration in animals. |
PC-42583 |
SKF 82958
Dopamine D1 agonist, ERα agonist
|
SKF 82958 is a potent, full dopamine D1 agonist, produces characteristic anorectic effects, hyperactivity and self-administration in animals. |
PC-45204 |
Metoclopramide
D2R antagonist
|
Metoclopramide is apotent dopamine D2 receptor antagonist with Ki of 28 nM. |
PC-42716 |
SB-277011
Dopamine D3 antagonist
|
SB-277011 is a potent and selective dopamine D3 receptor antagonist with pKi of 8.0. |
PC-22633 |
FOB02-04
D3R agonist
|
FOB02-04 is a potent, selective dopamine D3 receptor (D3R) agonist with Ki of 2.84 nM, weak affinity with Ki of 106 nM for D2R. |
PC-22235 |
Raclopride
Dopamine D2/D3 antagonist
|
Raclopride (FLA 870) is a potent, selective dopamine D2/D3 receptor antagonist, binds to D2 and D3 receptors with Ki of 1.8 nM and 3.5 nM, respectively. |
PC-22227 |
A-77636 hydrochloride
Dopamine D1 agonist
|
A-77636 hydrochloride is a potent, selective, orally active and long acting dopamine D1 receptor agonist with Ki of 39.8 nM. |