You are here:Home-Chemical Inhibitors & Agonists-GPCR-Dopamine Receptor

Request The Product List ofDopamine Receptor Dopamine Receptor

Cat. No. Product Name Information
PC-70062

ABT-724 trihydrochloride

Dopamine D4 agonist

ABT-724 trihydrochloride is a potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors.
PC-70061

ABT-724

Dopamine D4 agonist

A potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors.
PC-70057

PF-219061

PF-219061 (PF 219061, PF219061) is a potent, selective agonist of dopamine D3 receptor with EC50 of 8 nM.
PC-42584

SKF-82958 hydrobromide

Dopamine D1 agonist, ERα agonist

SKF-82958 hydrobromide is a potent, full dopamine D1 agonist, produces characteristic anorectic effects, hyperactivity and self-administration in animals.
PC-42583

SKF 82958

Dopamine D1 agonist, ERα agonist

SKF 82958 is a potent, full dopamine D1 agonist, produces characteristic anorectic effects, hyperactivity and self-administration in animals.
PC-45204

Metoclopramide

D2R antagonist

Metoclopramide is apotent dopamine D2 receptor antagonist with Ki of 28 nM.
PC-42716

SB-277011

Dopamine D3 antagonist

SB-277011 is a potent and selective dopamine D3 receptor antagonist with pKi of 8.0.
PC-22235

Raclopride

Dopamine D2/D3 antagonist

Raclopride (FLA 870) is a potent, selective dopamine D2/D3 receptor antagonist, binds to D2 and D3 receptors with Ki of 1.8 nM and 3.5 nM, respectively.
PC-22227

A-77636 hydrochloride

Dopamine D1 agonist

A-77636 hydrochloride is a potent, selective, orally active and long acting dopamine D1 receptor agonist with Ki of 39.8 nM.
PC-22147

SCH23390 hydrochloride

Dopamine Receptor antagonist

SCH23390 hydrochloride is a potent and selective dopamine D1-like receptor antagonist with Kis of 0.2 nM and 0.3 nM for the D1 and D5 receptor, respectively.
PC-21488

NGD-94-1

D4R inhibitor

NGD-94-1 is a highly potent, selective dopamine D4 receptor antagonist with Ki of 3.6 nM.
PC-21487

Nemonapride

D2R antagonist

Nemonapride (YM-09151-2) is a highly potent, selective dopamine D2 receptor antagonist with Ki of 0.06 nM.

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com