| Cat. No. |
Product Name |
Information |
| PC-21181 |
Ansofaxine
Triple reuptake inhibitor
|
Toludesvenlafaxine (Ansofaxine, LY03005, LPM570065) is a first-in-class triple monoaminergic reuptake inhibitor (TRI), blocks the reuptake of serotonin, dopamine, and norepinephrine with IC50 of of 723, 491 and 763 nM, respectively. |
| PC-21114 |
D-578
Monoamine reuptake inhibitor
|
D-578 is a potent, orally active triple monoamine reuptake inhibitor with Ki values of 16.2. 16.2, 3.23 nM, and 29.6, 20.6, 6.10 nM for the rat brain and cloned human dopamine, serotonin and norepinephrine transporters, respectively. |
| PC-20766 |
ZINC000443438219
SERT inhibitor
|
ZINC000443438219 (Compound 8219) is a highly potent, selective and non-competitive inhibitor of serotonin transporter (SERT) with Ki of 3 nM. |
| PC-20765 |
ZINC000006658090
SERT inhibitor
|
ZINC000006658090 (Compound 8090) is a highly potent, selective and non-competitive inhibitor of serotonin transporter (SERT) with Ki of 14 nM. |
| PC-20070 |
JJC8-091
DAT inhibitor
|
JJC8-091 is a potent, Modafinil-derived dopamine transporter (DAT) ligand / inhibitor with Ki of 16.7 nM, attenuates compulsive-like methamphetamine self-administration in rats. |
| PC-20069 |
JJC8-016
DAT ligand
|
JJC8-016 is a potent, Modafinil-derived dopamine transporter (DAT) ligand with Ki of 116 nM, attenuates compulsive-like methamphetamine self-administration in rats. |
| PC-20068 |
JJC8-088
DAT ligand
|
JJC8-088 is a potent, Modafinil-derived dopamine transporter (DAT) ligand / inhibitor with Ki of 2.53 nM. |
| PC-20035 |
FFN200 dihydrochloride
VMAT2 fluorescent
|
FFN200 dihydrochloride is a vesicular monoamine transporter 2 (VMAT2) substrate, and the first probe to selectively trace monoamine exocytosis in both neuronal cell culture and brain tissue. |
| PC-20034 |
FFN200
Fluorescent false neurotransmitter
|
FFN200 is a vesicular monoamine transporter 2 (VMAT2) substrate, and the first probe to selectively trace monoamine exocytosis in both neuronal cell culture and brain tissue. |
| PC-49734 |
NBI-98782
VMAT2 inhibitor
|
NBI-98782 (RRR-dihydrotetrabenazine, RRR-DHTBZ, (+)-α-HTBZ) is a potent, highly selective VMAT2 inhibitor (Ki=2 nM) and tetrabenazine metabolite. |
| PC-49497 |
SRI-20041
DAT inhibitor
|
SRI-20041 is a small molecule allosteric dopamine transporter ligand. |
| PC-49495 |
SRI-32743
DAT inhibitor
|
SRI-32743 is a novel allosteric modulator of dopamine transporter (DAT), attenuates HIV-1 Tat protein-induced inhibition of the dopamine transporter. |
