Cat. No. |
Product Name |
Information |
PC-43399 |
Vanoxerine dihydrochloride
Dopamine transport inhibitor
|
Vanoxerine (GBR-12909, I-893, Boxeprazine) is a highly potent inhibitor of dopamine uptake in vitro in tissue slices obtained from rat neostriatum with IC50 of 40-50 nM, also inhibits norepinephrine uptake with IC50 of 560-2600 nM. |
PC-63053 |
Atomoxetine hydrochloride
NET inhibitor
|
Atomoxetine hydrochloride((R)-Tomoxetine LY-139603) is a potent, selective norepinephrine (NE) transporter inhibitor with Ki of 5 nM. |
PC-63052 |
Atomoxetine
NET inhibitor
|
Atomoxetine ((R)-Tomoxetine, LY-139603) is a potent, selective norepinephrine (NE) transporter inhibitor with Ki of 5 nM. |
PC-62373 |
FFN-206 dihydrochloride
VMAT2 inhibitor
|
FFN-206 is an excellent VMAT2 (vesicular monoamine transporter 2) substrate capable of detecting VMAT2 activity in intact cells using fluorescence microscopy, with subcellular localization to VMAT2-expressing acidic compartments without apparent labeling of other organelles. |
PC-61998 |
Edivoxetine hydrochloride
Norepinephrine reuptake inhibitor
|
Edivoxetine (LY2216684) is a novel potent, selective norepinephrine reuptake inhibitor (NERI) being evaluated as adjunctive treatment for major depressive disorder (MDD). |
PC-61997 |
Edivoxetine
Norepinephrine reuptake inhibitor
|
Edivoxetine (LY2216684) is a novel potent, selective norepinephrine reuptake inhibitor (NERI) being evaluated as adjunctive treatment for major depressive disorder (MDD).. |
PC-61884 |
PF-184298
Monoamine reuptake inhibitor
|
PF-184298 is a potent, selective dual serotonin and noradrenaline monoamine reuptake inhibitor (SNRI) with IC50 of 6 nM and 21 nM, respectively. |
PC-70169 |
Amitifadine
Monoamine reuptake inhibitor
|
Amitifadine (DOV-21947, EB-1010) is a triple monoamine reuptake inhibitor, inhibits the reuptake of 5-HT, norepinephrine and dopamine in HEK 293 cells with IC50 of 12, 23 and 96 nM, respectively. |
PC-60053 |
Solriamfetol hydrochloride
|
Solriamfetol hydrochloride (JZP-110, R-228060, ADX-N05, YKP-10A) is a norepinephrine-dopamine reuptake inhibitor that inhibits dopamine and norepinephrine transporter with IC50 of 2.9 and 4.4 uM, respectively. |
PC-45481 |
Diclofensine
Monoamine reuptake inhibitor
|
Diclofensine (Ro 8-4650) is an antidepressant that acts as a triple monoamine reuptake inhibitor. |
PC-45480 |
Diclofensine hydrochloride
Monoamine reuptake inhibitor
|
Diclofensine (Ro 8-4650) hydrochloride is an antidepressant that acts as a triple monoamine reuptake inhibitor. |
PC-46649 |
Paroxetine hydrochloride
GRK2 inhibitor, SSRI
|
Paroxetine hydrochloride is an oral, selective serotonin reuptake inhibitor (SSRI), also is a direct, selective inhibitor of G protein-coupled receptor kinase 2 (GRK2) with pIC50 of 5.6. |