Cat. No. |
Product Name |
Information |
PC-20510 |
AT-076
Pan opioid antagonist
|
AT-076 (AT076) is the first potent small-molecule opioid pan antagonist with receptor binding Ki values of 1.75, 1.14, 1.67 and 19.6 nM for NOP, KOP, MOP, and DOP, respectively. |
PC-47497 |
D-Ala2, D-Leu5-Enkephalin
|
An angiotensin II analog that is an agonist of AT1 angiotensin receptor.. |
PC-45976 |
Alvimopan monohydrate
|
A selective peripherally acting μ-opioid antagonist with IC50 of 1.7 nM for the treatment of postoperative ileus. |
PC-45978 |
Naltrexone hydrochloride
|
A potent, competitive antagonist for μ, κ, δ, and σ-opioid receptors with Ki of 0.0825 nM, 0.509 nM, and 8.02 nM, for MOR, KOR, and DOR, respectively. |
PC-45960 |
Methylnaltrexone bromide
|
A peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.. |