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Cat. No. Product Name Information
PC-20510

AT-076

Pan opioid antagonist

AT-076 (AT076) is the first potent small-molecule opioid pan antagonist with receptor binding Ki values of 1.75, 1.14, 1.67 and 19.6 nM for NOP, KOP, MOP, and DOP, respectively.
PC-47497

D-Ala2, D-Leu5-Enkephalin

An angiotensin II analog that is an agonist of AT1 angiotensin receptor..
PC-45976

Alvimopan monohydrate

A selective peripherally acting μ-opioid antagonist with IC50 of 1.7 nM for the treatment of postoperative ileus.
PC-45978

Naltrexone hydrochloride

A potent, competitive antagonist for μ, κ, δ, and σ-opioid receptors with Ki of 0.0825 nM, 0.509 nM, and 8.02 nM, for MOR, KOR, and DOR, respectively.
PC-45960

Methylnaltrexone bromide

A peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals..

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