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Request The Product List ofOpioid Receptor Opioid Receptor

Cat. No. Product Name Information
PC-62107

Enadoline

KOR agonist

Enadoline (CI 977, PD 129290) is a potent, selective κ-opioid receptor (KOR) agonist with Ki of 0.11 nM, binding with high affinity to [3H]-U69593-labelled kappa-sites.
PC-61887

Spiradoline mesylate

KOR agonist

Spiradoline (U 62066) is a potent, highly selective κ-opioid agonist that has analgesic diuretic and antitussive effects..
PC-61886

Spiradoline

KOR agonist

Spiradoline (U 62066) is a potent, highly selective κ-opioid agonist that has analgesic diuretic and antitussive effects.
PC-61682

Oliceridine hydrochloride

MOR agonist

Oliceridine hydrochloride (Olinvo, TRV130) is a potent, selective, and G protein biased μ opioid receptor (MOR) agonist with pEC50 of 8.1.
PC-61681

Oliceridine

MOR agonist

Oliceridine (Olinvo, TRV130) is a potent, selective, and G protein biased μ opioid receptor (MOR) agonist with pEC50 of 8.1.
PC-61596

SR-8993

NOP-R agonist

SR-8993 is a potent, highly selective, brain-penetrant NOP-R (Nociceptin/orphanin FQ receptor) agonist with EC50 of 8.8 nM.
PC-61588

MK-1925

ORL1 agonist

MK-1925 is a selective, orally active, brain-penetrant opioid receptor-like 1 (ORL1.
PC-61550

AT-127

NOP receptor agonist

AT-127 is a potent, selective nociceptin/orphanin FQ receptor (NOP receptor) agonist with Ki of 1.18 nM.
PC-61549

AT-090

NOP receptor agonist

AT-090 is a potent, selective nociceptin/orphanin FQ receptor (NOP receptor) agonist with Ki of 5.61 nM.
PC-61547

SB-612111

NOP receptor antagonist

SB-612111 is a potent, selective nociceptin/orphanin FQ receptor (NOP receptor) antagonist with Ki of 0.33 nM.
PC-61546

LY2940094

NOP receptor antagonist

LY2940094 (BTRX246040) is a potent, selective, CNS-penetrant, orally available NOP (Nociceptin/OFQ) receptor antagonist with Kb of 0.17 nM.
PC-61545

J-113397

NOP antagonist

J-113397 is a potent, selective nociceptin/orphanin FQ receptor (NOP receptor/ORL1) antagonist with IC50 of 2.3 nM.

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