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Request The Product List ofOpioid Receptor Opioid Receptor

Cat. No. Product Name Information
PC-61536

SR16435

NOP/MOR agonist

SR16435 is a mixed NOP/μ-opioid partial agonist with equally high affinity (Ki=29 nM) for both NOP and μ-opioid receptors.
PC-70351

TAN-67 dihydrobromide

δ-opioid receptor agonist

TAN-67 dihydrobromide (SB205607) is a potent and selective δ-opioid receptor agonist that has high affinity and selectivity for the δ1 subtype with Ki of 1.12 nM.
PC-70350

KNT-127

DOR agonist

KNT-127 is a potent, selective δ-opioid receptor (DOR) agonist with Ki of 0.16 nM, dispalys 133.5-fold and 960.5-fold selectivity over μOR and κOR respectively.
PC-70349

SNC80

δ-opioid receptor agonist

SNC80 (NIH-10815) is a highly selective, non-peptide agonist of the δ-opioid receptor (δ-OR) with IC50/Ki of 2.73/0.18 nM.
PC-60804

TRV0109101

MOR agonist

TRV0109101 is a selective, G protein-biased µ-opioid receptor (MOR) agonist, does not promote the development of opioid-induced mechanical allodynia (OIMA) and rapidly reverses allodynia in vivo.
PC-60803

TRV0109101 hydrochloride

MOR agonist

TRV0109101 hydrochloride is a selective, G protein-biased µ-opioid receptor agonist, does not promote the development of opioid-induced mechanical allodynia (OIMA) and rapidly reverses allodynia in vivo.
PC-60802

NKTR-181

MOR agonist

A novel, long-acting and orally active, selective mu-opioid agonist that displays higher binding affinity (Ki=237 nM) at the MOR than kappa and delta opioid receptors (>100-fold).
PC-60800

SB-612111 hydrochloride

NOP receptor antagonist

SB-612111 hydrochloride is a potent, selective opiate receptor-like orphan receptor (ORL-1, NOP) antagonist with Ki of 0.33 nM.
PC-60799

AT-403

NOP agonist

AT-403 (AT403) is a potent, highly selective, nonpeptide NOP agonist with pEC50 of 9.45.
PC-60798

SCH 486757

ORL1 agonist

SCH 486757 is a potent, selective, orally active nociceptin/orphanin FQ peptide (NOP, ORL1) receptor agonist with Ki of 4.6 nM, with high selectiivity over classical opioid receptors.
PC-60797

SCH221510

NOP receptor agonist

SCH221510 is a potent, selective, orally active nociceptin opioid receptor (NOP) agonist with EC50 of 12 nM, Ki of 0.3 nM.
PC-60737

Eluxadoline

μ-opioid receptor agonist

A potent, selective, orally bioavailable µ-opioid receptor agonist and a δ-opioid receptor antagonist for the treatment of diarrhoea-predominant irritable bowel syndrome (IBS-D)..

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