| Cat. No. |
Product Name |
Information |
| PC-45979 |
Naltrexone
Opioid receptor antagonist
|
Naltrexone is a potent, competitive antagonist for μ, κ, δ, and σ-opioid receptors with Ki of 0.0825 nM, 0.509 nM, and 8.02 nM, for MOR, KOR, and DOR, respectively. |
| PC-45978 |
Naltrexone hydrochloride
Opioid receptor antagonist
|
Naltrexone hydrochloride is a potent, competitive antagonist for μ, κ, δ, and σ-opioid receptors with Ki of 0.0825 nM, 0.509 nM, and 8.02 nM, for MOR, KOR, and DOR, respectively. |
| PC-45960 |
Naltrexone methylbromide
Opioid receptor antagonist
|
Naltrexone methylbromide (Naltrexone methylbromide) is a peripherally-acting μ-opioid antagonist that acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals. |
| PC-45285 |
Meptazinol
MOR agonist
|
Meptazinol (IL-22811, WY-22811) is a partial µ-opioid receptor (MOR) agonist. |
| PC-42615 |
JDTic dihydrochloride
KOR antagonist
|
JDTic dihydrochloride is a highly potent and selective kappa Opioid receptor (KOR) antagonist with Ki of 0.3 nM. |
| PC-42614 |
JDTic
KOR antagonist
|
JDTic is a highly potent and selective kappa opioid receptor (KOR) antagonist with Ki of 0.3 nM. |
| PC-47491 |
Dynorphin A(1-13)
Neurolysin inhibitor, KOR agonist
|
Dynorphin A(1-13) is a potent, competitive peptidie inhibitor of Neurolysin (Nln) with IC50 of 1.2 uM, also is a kappa receptor agonist binds to human kappa opioid receptor (KOR) with Ki of 200 nM. |
| PC-27557 |
Naloxone hydrochloride
Opioid receptor antagonist
|
Naloxone hydrochloride is an opioid receptor antagonist, alleviates opioid-overdose-induced respiratory depression. |
| PC-27556 |
Naloxone
Opioid receptor antagonist
|
Naloxone is an opioid receptor antagonist, alleviates opioid-overdose-induced respiratory depression. |
| PC-27543 |
AT-324
MOP/NOP agonist
|
AT-324 is a potent, bifunctional agonist of nociceptin/orphanin FQ peptide (NOP/MOP) receptor with Ki of 1.28/1.46 nM, respectively. |
| PC-27542 |
AT-034
MOP/NOP agonist
|
AT-034 is a potent, bifunctional partial agonist of nociceptin/orphanin FQ peptide (NOP/MOP) receptor with Ki of 76.6 nM/1.97 nM, respectively. |
| PC-27541 |
AT-201
MOP/NOP agonist
|
AT-201 is a potent, bifunctional partial agonist of nociceptin/orphanin FQ peptide (NOP/MOP) receptor with Ki of 5.36 nM/2.7 nM, respectively. |
