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Cat. No. Product Name Information
PC-61544

Ro 64-6198

NOP agonist

Ro 64-6198 is a nonpeptidic, selective, brain-penetrant agonist of nociceptin/orphanin FQ receptor (NOP receptor/ORL1) with pKi of 9.41.
PC-61543

Ro 64-6198 hydrochloride

ORL1 agonist

Ro 64-6198 hydrochloride is a nonpeptidic, selective, brain-penetrant agonist of nociceptin/orphanin FQ receptor (NOP receptor/ORL1) with pKi of 9.41.
PC-61542

MT-7716

ORL1 agonist

A highly potent, brain-penetrating ORL1 receptor (NOP receptor) agonist with Ki of 0.76 and 0.50  nM for rat and human ORL1 receptors, respectively.
PC-61541

W-212393

ORL1 agonist

W-212393 (MT-7716 free base) is a highly potent, brain penetrant ORL1 receptor (NOP receptor) agonist with Ki of 0.76 and 0.50  nM for rat and human ORL1 receptors, respectively.
PC-61540

SR-16835

NOP receptor agonist

SR-16835 is a potent full agonist of ORL1 receptor (NOP receptor) with binding Ki of 11.4 nM, with low-affinity mu-opioid partial agonist activity (Ki=79.9 nM).
PC-61539

SR-16507

ORL1 agonist

SR-16507 is a potent full agonist of ORL1 receptor (NOP receptor) and partial agonist of mu-opioid receptor with Ki of 5.22 nM and 1.07 nM, respectively.
PC-61538

SR-16430

ORL1 inhibitor

SR-16430 is a selective ORL1 receptor (NOP receptor) antagonist that has 10-fold selectivity over μ-opioid receptor.
PC-61537

SR-14150

NOP/MOR agonist

SR-14150 is a potent NOP/μ-opioid partial agonist with Ki of 1.39 nM and 29.9 nM, respectively.
PC-61536

SR16435

NOP/MOR agonist

SR16435 is a mixed NOP/μ-opioid partial agonist with equally high affinity (Ki=29 nM) for both NOP and μ-opioid receptors.
PC-70351

TAN-67 dihydrobromide

δ-opioid receptor agonist

TAN-67 dihydrobromide (SB205607) is a potent and selective δ-opioid receptor agonist that has high affinity and selectivity for the δ1 subtype with Ki of 1.12 nM.
PC-70350

KNT-127

δ-opioid receptor agonist

KNT-127 is a potent, selective δ-opioid receptor (DOR) agonist with Ki of 0.16 nM, dispalys 133.5-fold and 960.5-fold selectivity over μOR and κOR respectively.
PC-70349

SNC80

δ-opioid receptor agonist

SNC80 (NIH-10815) is a highly selective, non-peptide agonist of the δ-opioid receptor (δ-OR) with IC50/Ki of 2.73/0.18 nM.

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