| Cat. No. |
Product Name |
Information |
| PC-61549 |
AT-090
|
AT-090 is a novel potent, selective nociceptin/orphanin FQ receptor (NOP receptor) agonist with Ki of 5.61 nM. |
| PC-61548 |
SB-612111 hydrochloride
|
SB-612111 is a potent, selective nociceptin/orphanin FQ receptor (NOP receptor) antagonist with Ki of 0.33 nM. |
| PC-61547 |
SB-612111
|
SB-612111 is a potent, selective nociceptin/orphanin FQ receptor (NOP receptor) antagonist with Ki of 0.33 nM. |
| PC-61546 |
LY-2940094
|
LY-2940094 (BTRX 246040) is a novel potent, selective, CNS-penetrant, orally available NOP (Nociceptin/OFQ) receptor antagonist with Kb of 0.17 nM. |
| PC-61537 |
SR-14150
|
SR-14150 is a potent NOP/μ-opioid partial agonist with Ki of 1.39 nM and 29.9 nM, respectively. |
| PC-61536 |
SR-16435
|
SR-16435 is a mixed NOP/μ-opioid partial agonist with equally high affinity (Ki=29 nM) for both NOP and μ-opioid receptors. |
| PC-70351 |
TAN-67 dihydrobromide
|
A potent and selective δ-opioid receptor agonist that has high affinity and selectivity for the δ1 subtype with Ki of 1.12 nM. |
| PC-60804 |
TRV0109101
|
A selective, G protein-biased µ-opioid receptor agonist, does not promote the development of opioid-induced mechanical allodynia (OIMA) and rapidly reverses allodynia in vivo.. |
| PC-60803 |
TRV0109101 hydrochloride
|
A selective, G protein-biased µ-opioid receptor agonist, does not promote the development of opioid-induced mechanical allodynia (OIMA) and rapidly reverses allodynia in vivo.. |
| PC-60800 |
SB-612111 hydrochloride
|
A potent, selective opiate receptor-like orphan receptor (ORL-1, NOP) antagonist with Ki of 0.33 nM. |
| PC-60797 |
SCH 221510
|
A potent, selective, orally active nociceptin opioid receptor (NOP) agonist with EC50 of 12 nM, Ki of 0.3 nM. |
| PC-60717 |
TK05
|
A potent and selective inhibitors of leukotriene C4 synthase (LTC4S) with IC50 of 95 nM, Ki of 6 nM. |
