Cat. No. |
Product Name |
Information |
PC-42894 |
Umeclidinium bromide
|
Umeclidinium bromide (GSK 573719A) is potent, long-acting, inhaled antagonist of mAChRs with Ki of 0.05-0.16 nM for human M1-M5 mAChRs. |
PC-62144 |
ML381 fumarate
|
ML381 (VU0488130) is a highly mAChR subtype selective M5 orthosteric antagonist with IC50/Ki of 450/340 nM for hM5, has no inhibitory activity on hM1-4 (IC50>30 uM). |
PC-61893 |
Fesoterodine fumarate
|
Fesoterodine (PF-00695838) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties. |
PC-61892 |
Fesoterodine maleate
|
Fesoterodine (PF-00695838) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties. |
PC-61761 |
Glycopyrronium bromide
|
Glycopyrronium bromide (CHF 5259) is a peripherally-acting quaternary ammonium antimuscarinic agent with little or no central nervous system activity. |
PC-42262 |
Pirmenol hydrochloride
|
An orally effective, long-acting antiarrhythmic agent that interacts with cardiac muscarinic receptors.. |
PC-45938 |
Cevimeline
|
A potent M1-selective muscarinic agonist. |
PC-45283 |
Glycopyrrolate
|
A muscarinic anticholinergic that blocks muscarinic receptors, thus inhibiting cholinergic transmission.. |
PC-45180 |
Tiotropium bromide
|
A long-acting muscarinic receptor antagonist that used in the management of chronic obstructive pulmonary disease (COPD).. |