You are here:Home-Chemical Inhibitors & Agonists-PI3K/Akt/mTOR Pathway-PI3K

Request The Product List ofPI3K PI3K

Cat. No. Product Name Information
PC-42925

PI-3065

p110δ inhibitor

PI-3065 is a potent inhibitor of PI3K p110δ with IC50/Ki values of 5/1.5 nM respectively.
PC-45869

ZSTK-474

PI3K inhibitor

ZSTK-474 (ZSTK474) is a potent inhibitor of class I PI3K isoforms with IC50 of 17 nM, 53 nM, and 6 nM for p110β, p110γ, and p110δ, respectively.
PC-42695

PKI-402

PI3K/mTOR inhibitor

PKI-402 is a potent dual PI3K/mTOR inhibitor with IC50 of 1/7/16/14/1.7 nM for PI3Kα/β/γ/δ/mTOR respectively.
PC-42315

IC-87114

PI3Kδ inhibitor

IC-87114 (IC87114) is a potent and selective PI3Kδ inhibitor with IC50 of 0.5 uM.
PC-42326

SF2523

PI3K/BRD4 inhibitor

SF2523 is a potent, dual inhibitor of PI3K and BRD4 with IC50 of 241, 34, 158 nM for BRD4 (BD1), PI3Kα and PI3Kγ, respectively.
PC-45394

Leniolisib

PI3Kδ inhibitor

Leniolisib (CDZ173) is a potent and selective PI3Kδ inhibitor with biochemical IC50 of 11 nM.
PC-42518

PIK-294

p110δ inhibitor

PIK-294 is a highly potent, selective p110δ inhibitor with IC50 of 10 nM, shows 1000-, 49- and 16-fold less potent to PI3Kα/β/γ.
PC-42513

Omipalisib

PI3K/mTOR inhibitor

Omipalisib (GSK2126458) is a highly potent dual inhibitor PI3K/mTOR inhibitor with app Ki of 19/130/24/60/180/300 nM for p110α/p110β/p110γ/p110δ/mTORC1/mTORC2 respectively.
PC-42133

PF-04979064

PI3K/mTOR inhibitor

PF-04979064 is a highly potent and selective, dual PI3K/mTOR inhibitor with Ki of 0.13, 0.111, 0.122 and 1.42 nM for PI3Kα, PI3Kγ, PI3Kδ and mTOR, respectively.
PC-42310

LY294002

PI3K inhibitor

LY294002 is a classic, broad-spectrum PI3K inhibitor with IC50 of 0.5/0.57/0.97 uM for PI3Kα/δ/β, respectively.
PC-21948

PIK-108

p110β inhibitor

PIK-108 is a potent, selective and allosteric PI3K p110β inhibitor with IC50 of 57 nM, 45-fold selective over PI3Kα (IC50=2600 nM).
PC-21947

PI3Kα H1047R inhibitor 17

H1047R PI3Kα inhibitor

PI3Kα H1047R inhibitor 17 is a potent, selective H1047R PI3Kα mutant inhibitor with IC50 of 1 nM (inhibition of pAKT formation), without effect on PI3Kα WT.

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com