| Cat. No. |
Product Name |
Information |
| PC-42340 |
AZD1152-HQPA
Aurora B inhibitor
|
AZD1152-HQPA (Barasertib-HQPA, AZD2811) is the active product of AZD1152, a potent, selective inhibitor of Aurora B kinase with IC50 of 0.37 nM. |
| PC-42424 |
MLN8054
Aurora A inhibitor
|
MLN8054 (MLN-8054) is a potent, selective, ATP-competitive, orally active Aurora A kinase inhibitor with IC50 of 4 nM. |
| PC-45943 |
GSK1070916
Aurora B/C inhibitor
|
GSK1070916 (GSK-1070916A) is a potent, selective and ATP-competitive inhibitor of Aurora B and Aurora C with Ki of 0.38 nM and 1.5 nM, respectively. |
| PC-42612 |
SCH-1473759 hydrochloride
Aurora A/B inhibitor
|
SCH-1473759 hydrochloride is a potent, picomolar, dual inhibitor of Aurora A and Aurora B with IC50 of 0.02 and 0.03 nM, respectively. |
| PC-42611 |
SCH-1473759
Aurora A/B inhibitor
|
SCH-1473759 is a potent, picomolar, dual inhibitor of Aurora A and Aurora B with IC50 of 0.02 and 0.03 nM, respectively. |
| PC-42703 |
CCT 137690
Aurora Kinase inhibitor
|
CCT 137690 is a potent, orally bioavailable Aurora kinases inhibitor with IC50 of 15/25/19 nM for Aurora A/B/C, respectively. |
| PC-42420 |
PHA-680632
Aurora Kinase inhibitor
|
PHA-680632 is a potent, highly selective Aurora kinase inhibitor with IC50 of 27, 135 and 120 nM for Aurora A, B and C, respectively. |
| PC-42342 |
Barasertib
Aurora B inhibitor
|
Barasertib (AZD1152) is a potent, highly selective Aurora B inhibitor with IC50 of 0.37 nM. |
| PC-45948 |
TCS7010
Aurora A inhibitor
|
TCS7010 is a potent, highly selective Aurora A inhibitor with IC50 of 3.4 nM. |
| PC-42422 |
Danusertib
Aurora kinase inhibitor
|
Danusertib (PHA-739358) is a potent, ATP-competitive Aurora kinase inhibitor with IC50 of 13,79 and 61 nM for Aurora A, B and C, respectively. |
| PC-42650 |
CYC-116
Aurora A/B inhibitor
|
CYC-116 (CYC116) is a potent and selective Aurora A/Aurora B inhibitor with IC50 of 8.0/9.2 nM. |
| PC-42757 |
Alisertib
Aurora A inhibitor
|
Alisertib (MLN8237) is a potent and highly selective inhibitor of Aurora A (AURKA) with IC50 of 1.2 nM. |
