| Cat. No. |
Product Name |
Information |
| PC-20472 |
IU1-206
USP14 inhibitor
|
IU1-206 is a IU1 derivative with more potent activity against USP14, 10-fold more potent than IU1 and is comparable to the IU1-47. |
| PC-20403 |
PR-619
DUBs inhibitor
|
PR-619 (PR619) is a broad-spectrum, reversible deubiquitinating enzymes (DUBs) inhibitor with IC50 of 3.93 uM-8.87 uM. |
| PC-20202 |
HBX41108
USP7 inhibitor
|
HBX41108 is a specific small-molecule inhibitor of USP7/HAUSP ubiquitin protease with IC50 of 424 nM for inhibition of Ub-AMC hydrolysis by USP7. |
| PC-20190 |
USP14 inhibitor 3
USP14 inhibitor
|
USP14-IN-3 is a specific small molecule USP14 inhibitor with IC50 of <0.5 uM. |
| PC-20189 |
USP14 inhibitor 2
USP14 inhibitor
|
USP14-IN-2 is a specific small molecule USP14 inhibitor with IC50 of <0.5 uM. |
| PC-20186 |
USP14 inhibitor 1
USP14 inhibitor
|
USP14-IN-1 is a specific small molecule USP14 inhibitor with IC50 of 0.5 uM. |
| PC-20185 |
IU2-6
USP14 inhibitor
|
IU2-6 is a small molecule USP14 inhibitor, shows 74% inhibition at 8 uM. |
| PC-20184 |
GSK2643943A
USP20 inhibitor
|
GSK2643943A is a specific, cell penetrant small molecule inhibitor of deubiquitinating enzyme USP20 with IC50 of 160 nM (USP20/Ub-Rho). |
| PC-20004 |
TG2-179-1
BAP1 inhibitor
|
TG2-179-1 is a potent, selective and covalently inhibitor of deubiquitinase (DUB) BRCA1-associated protein-1 (BAP1), covalently binds to the active site of BAP1 (Cys91), exhibits potent cytotoxic activity against colon cancer cells. |
| PC-20001 |
CAS-12290-201
VCPIP1 inhibitor
|
CAS-12290-201 is a potent and selective inhibitor of deubiquitinating enzyme (DUB) VCPIP1 with IC50 of 70 nM, covalently and specificly targets the catalytic cysteine of VCPIP1 with little to no activity toward other cellular DUBs. |
| PC-49863 |
BAY-728
BAY-805 negative control
|
BAY-728 (BAY728, (S)-BAY-805) is a less potent enantiomer and negative control compound of BAY-805, which is a potent and selective Inhibitor of USP21. |
| PC-49862 |
BAY-805
USP21 inhibitor
|
BAY-805 (BAY805) is the first highly potent, selective and non-covalent USP21 inhibitor with IC50 of 6 nM and 2 nM in HTRF and Ub-rhodamine biochemical assays (hUSP21), respectively. |
