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Cat. No. Product Name Information
PC-49401

SR10221

PPARγ inverse agonist

SR10221 is a potent, selective PPARγ inverse agonist with IC50 of 13 nM in biochemical peptide recruitment assays, represses downstream PPARγ target genes leading to growth inhibition in bladder cancer cell lines.
PC-49400

BAY-0069

PPARγ inverse agonist

BAY-0069 (BAY0069) is a potent, selective, covalent PPARγ inverse agonist with IC50 of 0.22 nM in cellular reporter assays.
PC-49036

GQ-16

PPARγ agonist

GQ-16 is a peroxisome proliferator-activated receptor γ (PPARγ) ligand and partial agonist with Ki value of 160 nM, specific for PPARγ with no detectable activity to activate other PPAR subtypes (PPARα or PPARβ/δ) or RXRα.
PC-73409

Bocidelpar

PPARδ agonist

Bocidelpar (ASP-0367, MA-0211, MTB-1) is a potent selective peroxisome proliferator-activated receptor delta (PPARδ) agonist with potential against mitochondrial myopathies.
PC-73019

MSDC0160

MPC inhibitor

MSDC0160 (Mitoglitazone, MSDC-0160) is a small molecule targeting mitochondrial pyruvate carrier (MPC), also is an insulin sensitizer with anti-diabetes activities.
PC-72950

PPARγ pSer273-IN-10

PPARγ pSer273 inhibitor

PPARγ pSer273-IN-10 is a specific, in vivo-active small molecule inhibitor of CDK5-mediated Ser273 phosphorylation of PPARγ without classical PPARγ agonism.
PC-38250

WO95E

PPARγ agonist

WO95E is a novel potent, synthetic ligand (partial agonist) of PPARγ, directly binds to PPARγ with IC50 of 11 nM.
PC-38051

EHP-101

EHP-101 (Etrinabdione, VCE-004.8) is an orally active, specific PPARγ and CB2 receptor dual agonist.
PC-35795

Chiglitazar

Chiglitazar (Carfloglitazar, CS-038, CS038) is a potent, dual PPARα/γ dual agonist with EC50 of 1.2, 0.08, 1.7 uM for PPARα, PPARγ and PPARδ, respectively.
PC-43387

T0070907

PPARγ inhibitor

T0070907 is a potent, selective, covalent PPARγ antagonist with binding IC50 of 1 nM, >800-fold preference for PPARγ over PPARα and PPARδ.
PC-62872

GW-6471

PPARα inhibitor

GW-6471 is a potent PPARα antagonist with IC50 of 0.24 uM, enhances the binding affinity of the PPARα ligand-binding domain to the co-repressor proteins SMRT and NCoR..
PC-61631

ABTL0812

ABTL0812 (2-hydroxylinoleic acid) is a novel first-in-class, small molecule that inhibits the Akt/mTORC1 axis and shows antiproliferative effect on tumor cells.

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