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Cat. No. Product Name Information
PC-42524

CL-387785

EGFR inhibitor

CL-387785 (EKI785, WAY-EKI785) is a specific, irreversible, covalent EGFR inhibitor with IC50 of 0.37 nM.
PC-42522

BIBX 1382

EGFR inhibitor

BIBX 1382 (Falnidamol) is a selective EGFR inhibitor with IC50 of 3 nM.
PC-45895

Lapatinib ditosylate

EGFR inhibitor

Lapatinib (GW 572016) ditosylate is a reversible, selective dual tyrosine kinase inhibitor of both EGFR and ErbB2 with IC50 of 10.8 and 9.2 nM in cell-free assays, respectively.
PC-45894

Lapatinib

EGFR inhibitor

Lapatinib (GW572016) is a reversible, selective dual tyrosine kinase inhibitor of both EGFR and ErbB2 with IC50 of 10.8 and 9.2 nM in cell-free assays, respectively.
PC-45997

AZD-9291 dimesylate

mutant EGFR inhibitor

Osimertinib dimesylate (AZD-9291) is a potent, selective, third-generation irreversible inhibitor of mutant EGFR with IC50s of 1/12/5 nM for L858R-T790M/L858R/L861Q respectively.
PC-44707

AZD-9291 mesylate

mutant EGFR inhibitor

Osimertinib mesylate (AZD-9291) is a potent, selective, third-generation irreversible inhibitor of mutant EGFR with IC50s of 1/12/5 nM for L858R-T790M/L858R/L861Q respectively. Osimertinib shows weak activity against wt EGFR (IC50=184 nM).
PC-44706

AZD-9291

mutant EGFR inhibitor

Osimertinib (AZD-9291) is a potent, selective, third-generation irreversible inhibitor of mutant EGFR with IC50s of 1/12/5 nM for L858R-T790M/L858R/L861Q respectively.
PC-45812

Pelitinib

EGFR inhibitor

Pelitinib (EKB-569, WAY-EKB 569) is a potent, selective, orally active, irreversible inhibitor of EGFR with IC50 of 80 nM.
PC-45892

Gefitinib hydrochloride

EGFR inhibitor

Gefitinib hydrochloride (ZD1839) is a potent, selective, orally active EGFR inhibitor with IC50 of 23 nM.
PC-45891

Gefitinib

EGFR inhibitor

Gefitinib (ZD1839) is a potent, selective, orally active EGFR inhibitor with IC50 of 23 nM.
PC-45893

Erlotinib

EGFR inhibitor

Erlotinib (OSI-744; R-1415; CP-358774) is a potent, selective inhibitor of EGFR with IC50 of 2 nM.
PC-42486

BMS-599626

EGFR/HER2 inhibitor

BMS-599626 (AC480) is a potent, selective inhibitor of EGFR and HER2 with IC50 of 20 nM and 30 nM.

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