| Cat. No. |
Product Name |
Information |
| PC-62304 |
HER2-IN-3
|
HER2-IN-3 is a type I HER2 inhibitor that has a similar profile to HER2-IN-2. |
| PC-62303 |
HER2-IN-2
|
HER2-IN-2 is a potent, selective HER2 inhibitor, only shows potent inhibition for EGFR and Abl in a panel of kinases. |
| PC-60540 |
FD-5180
|
A novel protein kinase affinity probe.. |
| PC-60378 |
SU-5214
|
A tyrosine kinase signal transduction modulator.. |
| PC-42641 |
ARRY-380 analog
|
An analog of ARRY-380, a potent and selective HER2 inhibitor with IC50 of 8 nM. |
| PC-45997 |
AZD-9291 dimesylate
|
A potent, selective, third-generation irreversible inhibitor of mutant EGFR with IC50s of 1/12/5 nM for L858R-T790M/L858R/L861Q respectively. |
| PC-44707 |
AZD-9291 mesylate
|
A potent, selective, third-generation irreversible inhibitor of mutant EGFR with IC50s of 1/12/5 nM for L858R-T790M/L858R/L861Q respectively. |
| PC-45892 |
Gefitinib hydrochloride
|
A potent, selective, orally active EGFR inhibitor with IC50 of 23 nM. |
| PC-44667 |
CO-1686 hydrobromide
|
A potent, highly selective, irreversible inhibitor of mutant EGFR with Ki of 21.5 nM for EGFR L858R/T790M. |
| PC-42386 |
RG13022
|
A potent EGFR inhibitor that inhibits EGFR autophosphorylation with IC50 of 5 uM in cell-free assays. |
| PC-42383 |
RG14620
|
A potent EGFR inhibitor that inhibits EGFR autophosphorylation with IC50 of 4 uM in cell-free assays. |
| PC-46002 |
O-Desmorpholinopropyl Gefitinib
|
A metabolite of Gefitinib, which is a potent inhibitor of tyrosine phosporylation in EGFR.. |
