| Cat. No. |
Product Name |
Information |
| PC-45033 |
Eltoprazine hydrochloride
5-HT1A/5-HT1B agonist
|
Eltoprazine hydrochloride (DU28853) is an antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor. |
| PC-45032 |
Eltoprazine
5-HT1A/5-HT1B agonist
|
Eltoprazine (DU-28853, DU28853) is an antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor. |
| PC-45212 |
Loxapine
D4/5-HT2 antagonist
|
Loxapine is a typical antipsychotic agent and D4/5-HT2 antagonist that displays an extremely strong binding affinity for dopamine D4 and serotonin 5-HT2 receptors. |
| PC-45797 |
Setiptiline
α2 adrenoceptor antagonist
|
Setiptiline (Teciptiline, Org8282, MO-8282) is a tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, as well as an H1 receptor inverse agonist/antihistamine. |
| PC-45034 |
RU 24969
5-HT1B agonist
|
RU 24969 is a potent, selective agonist of 5-HT1A and 5-HT1B receptors with Ki values of 2.5 and 0.38 nM respectively, with preference for 5-HT1B. |
| PC-42651 |
Nelotanserin
5-HT2A antagonist
|
Nelotanserin (RVT-102, APD125) is a potent, selective 5-HT2A inverse agonist with pKi of 9.2. |
| PC-45757 |
Eptapirone
5-HT1A agonist
|
Eptapirone (F11440) is a potent, selective 5-HT1A receptor agonist with Ki of 4.8 nM, pKi of 8.33. |
| PC-45945 |
Alosetron hydrochloride
5-HT3 antagonist
|
Alosetron (GR-68755) hydrochloride is a potent and selective 5-HT3 receptor antagonist has been shown to be beneficial in the treatment of irritable bowel syndrome. |
| PC-45944 |
Alosetron
5-HT3 antagonist
|
Alosetron (GR-68755) is a potent and selective 5-HT3 receptor antagonist has been shown to be beneficial in the treatment of irritable bowel syndrome. |
| PC-42547 |
WAY-100635
5-HT1A antagonist
|
WAY-100635 (WAY100635) is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor. |
| PC-42653 |
Ketanserin
5-HT2A antagonist
|
Ketanserin (R41468) is a high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C. |
| PC-45229 |
Ziprasidone hydrochloride monohydrate
D2/5-HT2A antagonist
|
Ziprasidone hydrochloride monohydrate (CP-88059) is a full antagonist of D2 and 5-HT2A receptors with Ki of 6.8 and 0.6 nM, respectively. |
