| Cat. No. |
Product Name |
Information |
| PC-73299 |
Usmarapride
5-HT4 agonist
|
Usmarapride (SUVN-D4010) is a potent, selective, orally active and brain penetrant 5-HT4 receptor partial agonist with EC50of 44 nM. |
| PC-35019 |
Ro 60-0175 fumarate
|
Ro 60-0175 is a potent, selective 5-HT2C receptor agonist with pKi of 9, 7.5, 5.4, 5.2 and 5.6 for human 5-HT2C, 2A, 1A, 6 and 7 receptors respectively. |
| PC-43384 |
BRL-15572 dihydrochloride
|
BRL-15572 is a potent, selective h5-HT1D receptor antagonist with pKi of 7.9, dispalys 60-fold selectivity over h5-HT1B. |
| PC-63186 |
DSP-6952 hydrobromide
|
DSP-6952 is a novel potent, selective, orally active 5-HT4 receptor partial agonist with Ki of 50-100 nM for human 5-HT4a/4b/4c. |
| PC-61503 |
AVN-322 free base
|
A highly selective, potent, BBB penetrant and orally bioavailable 5-HT6R antagonist for the treatment of neurological disorders such as AD and schizophrenia. |
| PC-60046 |
Landipirdine
|
A novel 5-HT receptor antagonist for the treatment of Parkinson's disease.. |
| PC-45693 |
Lumateperone tosylate
|
Lumateperone (ITI-007) is a potent 5-HT2A antagonist (Ki=0.54 nM), postsynaptic D2 antagonist(Ki=32 nM), and SERT blocker (Ki= 61 nM). |
| PC-45233 |
Iloperidone hydrochloride
|
An atypical antipsychotic that exhibits high affinity to serotonin 5HT2A (Ki =5.6 nM), dopamine D2 (Ki=6.3 nM) and D3 (Ki=7.1 nM) and noradrenaline α1 receptors (Ki=0.36 nM), moderate affinity for D4 (25 nM), 5HT6 (43 nM), 5HT7 (22 nM), and low affinity for 5HT1A (168 nM), D1 and histamine H1 receptors. |
| PC-42792 |
Risperidone mesylate
|
An antipsychotic agent with serotonin-S2 and dopamine-D2 antagonistic properties. |
| PC-42791 |
Risperidone hydrochloride
|
An antipsychotic agent with serotonin-S2 and dopamine-D2 antagonistic properties. |
| PC-42790 |
Risperidone
|
An antipsychotic agent with serotonin-S2 and dopamine-D2 antagonistic properties. |
| PC-45033 |
Eltoprazine hydrochloride
|
An antiaggressive agent that acts as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.. |
