| Cat. No. |
Product Name |
Information |
| PC-63186 |
DSP-6952 hydrobromide
|
DSP-6952 is a novel potent, selective, orally active 5-HT4 receptor partial agonist with Ki of 50-100 nM for human 5-HT4a/4b/4c. |
| PC-62934 |
Perlapine
|
Perlapine (AW-14233. |
| PC-62760 |
SB 206553
|
SB 206553 is a potent and selective 5-HT2B/5-HT2C receptor antagonist with pA2 of 8.89 for rat 5-HT2B, pKi of 7.92 for human 5-HT2C, displays >80-fold selectivity over other 5-HT receptor subtypes. |
| PC-62095 |
Velusetrag hydrochloride
|
Velusetrag (TD-5108) is a potent, selective and oral 5-HT4 receptor agonist with pKi of 7.7, shows >500-fold selectivity over other 5-HT receptors. |
| PC-62094 |
Velusetrag
|
Velusetrag (TD-5108) is a potent, selective and oral 5-HT4 receptor agonist with pKi of 7.7, shows >500-fold selectivity over other 5-HT receptors. |
| PC-62010 |
VA-012
|
VA-012 is a potent, selective 5-HT2C receptor positive allosteric modulator (PAM) that exhibits dose-dependent potentiation of 5-HT efficacy with EC50 of 16 nM. |
| PC-61868 |
Eletriptan
|
Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist. |
| PC-61867 |
Eletriptan hydrobromide
|
Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist. |
| PC-61814 |
SB 737050A
|
SB 737050A is a potent, selective 5-HT6 receptor antagonist to prevent relapse intio addiction.. |
| PC-61812 |
GSK-812
|
GSK-812 is a potent neuroprotectant that can induce GDNF in normal and diseased retina, shows has polypharmacology antagonizing multiple receptors, including D2 and D3 receptors, and 5-HT2A, 2C, and 5-HT6 receptors.. |
| PC-61729 |
Revexepride
|
Revexepride (SSP 002358. |
| PC-61583 |
GSK-588045
|
GSK-588045 is a potent and selective 5-HT1A/B/D receptor antagonist with Ki of 9.5/8.8/9.8, respectively. |
