| Cat. No. |
Product Name |
Information |
| PC-21048 |
NU-1223
5-HT2C agonist
|
NU-1223 is a β carboline analog of alstonine and serotonin 5-HT2C receptor agonist, blocks phencyclidine and amphetamine-induced hyperactivity in subchronic phencyclidine mice. |
| PC-20845 |
EMD386088 hydrochloride
5-HT6 agonist
|
EMD386088 hydrochloride is a potent, selective 5-HT6 receptor agonist with EC50 of 1.0 nM. |
| PC-20844 |
EMD386088
5-HT6 agonist
|
EMD386088 is a potent, selective 5-HT6 receptor agonist with EC50 of 1.0 nM. |
| PC-20843 |
SAM-531
5-HT6 agonist
|
SAM-531 (Cerlapirdine, WAY-262531) is a selective, highly potent, 5-HT6 receptor antagonist. |
| PC-38596 |
SB 224289 hydrochloride
5-HT1B antagonist
|
SB 224289 hydrochloride is a potent, selective 5-HT1B inverse agonist/antagonist with pKi value of 8.16, displays >75-fold selectivity over all other 5-HT receptors. |
| PC-45233 |
Iloperidone hydrochloride
|
An atypical antipsychotic that exhibits high affinity to serotonin 5HT2A (Ki =5.6 nM), dopamine D2 (Ki=6.3 nM) and D3 (Ki=7.1 nM) and noradrenaline α1 receptors (Ki=0.36 nM), moderate affinity for D4 (25 nM), 5HT6 (43 nM), 5HT7 (22 nM), and low affinity for 5HT1A (168 nM), D1 and histamine H1 receptors. |
| PC-42792 |
Risperidone mesylate
|
An antipsychotic agent with serotonin-S2 and dopamine-D2 antagonistic properties. |
| PC-42791 |
Risperidone hydrochloride
|
An antipsychotic agent with serotonin-S2 and dopamine-D2 antagonistic properties. |
| PC-45213 |
Loxapine succinate
|
A typical antipsychotic agent that displays an extremely strong binding affinity for dopamine D4 and serotonin 5-HT2 receptors.. |
| PC-45798 |
Setiptiline maleate
|
A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, as well as an H1 receptor inverse agonist/antihistamine.. |
| PC-42655 |
Sarpogrelate hydrochloride
|
A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A. |
| PC-43964 |
Ziprasidone hydrochloride
|
A full antagonist of D2 and 5-HT2A receptors with Ki of 6.8 and 0.6 nM, respectively. |
