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Cat. No. Product Name Information
PC-45757

Eptapirone

5-HT1A agonist

Eptapirone (F11440) is a potent, selective 5-HT1A receptor agonist with Ki of 4.8 nM, pKi of 8.33.
PC-42334

Asenapine

5-HT antagonist

Asenapine (Org5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors.
PC-45945

Alosetron hydrochloride

5-HT3 antagonist

Alosetron (GR-68755) hydrochloride is a potent and selective 5-HT3 receptor antagonist has been shown to be beneficial in the treatment of irritable bowel syndrome.
PC-45944

Alosetron

5-HT3 antagonist

Alosetron (GR-68755) is a potent and selective 5-HT3 receptor antagonist has been shown to be beneficial in the treatment of irritable bowel syndrome.
PC-42547

WAY-100635

5-HT1A antagonist

WAY-100635 (WAY100635) is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor.
PC-42654

Ketanserin tartrate

5-HT2A antagonist

Ketanserin tartrate (R41468 tartrate) is a high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.
PC-42653

Ketanserin

5-HT2A antagonist

Ketanserin (R41468) is a high-affinity, non-selective antagonist of 5-HT2 receptor with Ki of 2-3 nM for 5-HT2A and 28 nM for 5-HT2C.
PC-45229

Ziprasidone hydrochloride monohydrate

D2/5-HT2A antagonist

Ziprasidone hydrochloride monohydrate (CP-88059) is a full antagonist of D2 and 5-HT2A receptors with Ki of 6.8 and 0.6 nM, respectively.
PC-43963

Ziprasidone

D2/5-HT2A antagonist

Ziprasidone (CP 88059) is a full antagonist of D2 and 5-HT2A receptors with Ki of 6.8 and 0.6 nM, respectively.
PC-25204

Mirtazapine

5-HT antagonist

Mirtazapine (Org3770) is a potent and orally active 5-HT2, 5-HT3, histamine H1 receptor and α2-adrenoceptor antagonist with pKi values of 8.05, 8.1, 9.3 and 6.95, respectively, noradrenergic and specific serotonergic antidepressant (NaSSA) agent.
PC-25075

(S)-Hydroxy Iloperidone

CAS 501373-88-2

(S)-Hydroxy Iloperidone (Milsaperidone) is a metabolite of Iloperidone, which is an atypical antipsychotic, binds to adrenergic α1 and α2c receptors with pKi of 9.2 and 7.7 respectively.
PC-25028

Remlifanserin

5-HT2A inverse agonist

Remlifanserin is a potent, selective 5-HT2A serotonin receptor inverse agonist.

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