| Cat. No. |
Product Name |
Information |
| PC-60545 |
Arimoclomol maleate
|
Arimoclomol maleate (BRX-220) is a nontoxic, orally active heat shock protein (HSP) coinducer and potentiator of the heat shock response. |
| PC-60544 |
Arimoclomol
|
Arimoclomol (BRX-220) is a nontoxic heat shock protein (HSP) coinducer and potentiator of the heat shock response. |
| PC-60497 |
SM253
HSP90 inhibitor
|
SM253 (SM 253, SM-253) is a novel potent Hsp90 inhibitor that does not induce heat shock response. |
| PC-60471 |
MPC-3100
HSP90 inhibitor
|
MPC-3100 is a novel potent, selective, orally bioavailable Hsp90 inhibitor with IC50 of 0.14 uM. |
| PC-60470 |
MPC-0767
HSP90 inhibitor
|
MPC-0767 (MPC0767, MPC3100 mesylate hydrate) is an L-alanine ester prodrug of MPC-3100, which is a potent, selective, orally bioavailable Hsp90 inhibitor with IC50 of 0.14 uM. |
| PC-60233 |
CCT251236
Pirin ligand
|
CCT251236 (CCT-251236) is a potent, orally available Pirin ligand (Ki=28 nM), blocks the HSF1-mediated induction of both HSP72 and HSP27. |
| PC-60157 |
PU-H54
|
PU-H54 is a potent, selective Grp94 inhibitor. |
| PC-42460 |
PF-04929113 Mesylate
HSP90 inhibitor
|
The prodrug of PF-04928473 (SNX-2112), a potent, orally bioavailable HSP90 inhibitor. |
| PC-42456 |
Retaspimycin hydrochloride
HSP90 inhibitor
|
A water-soluble derivative of 17-AAG and HSP90 inhibitor. |
| PC-42156 |
HA-15
GRP78 inhibitor
|
HA-15 is a specifc inhibitor of the chaperone BiP (Binding immunoglobulin protein, GRP78 or HSPA5) that displays anti-cancerous activity on melanoma cells, including BRAF resistance melanoma cells. |
| PC-42278 |
KRIBB11
HSF1 inhibitor
|
KRIBB11 is a small molecule heat shock factor 1 (HSF1) inhibitor with IC50 of 1.2 uM. |
| PC-42459 |
BIIB021
HSP90 inhibitor
|
BIIB021 is a potent, selective, orally available HSP90 inhibitor with Ki of 1.7 nM for Hsp90α. |
