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Cat. No. Product Name Information
PC-42419

AMG-9810

TRPV1 inhibitor

AMG-9810 is a potent, selective and competitive TRPV1 antagonist with IC50 of 24.5 and 85.6 nM for human and rat TRPV1, respectively.
PC-45556

PF-4840154

TRPA1 agonist

PF-4840154 is a potent, selective agonist of the rat (EC50=97 nM) and human (EC50=23 nM) TRPA1 channel.
PC-42017

SKF-96365 hydrochloride

SOCE inhibitor

SKF-96365 hydrochloride (SKF96365) is potent inhibitor of receptor-mediated calcium entry (RMCE) with IC50 of 8.5 and 11.7 uM for inhibition in platelets stimulated with ADP and thrombin, respectively.
PC-42689

AMG517

TRPV1 antagonist

AMG517 is a potent and selective vanilloid receptor TRPV1 antagonist with IC50 of 0.76 nM for hTRPV
PC-42931

SB-366791

TRPV1 antagonist

SB-366791 (SB366791) is a potent and selective vanilloid receptor (VR1/TRPV1) antagonist with IC50 of 5.7 nM, also enhances oligodendrocyte formation via HSD17B7 inhibition.
PC-42084

HC-067047

TRPV4 inhibitor

HC-067047 (HC067047) is a potent and selective TRPV4 antagonist with IC50 of 48 nM, 133 nM, and 17 nM for human, rat, and mouse TRPV4 in cell assays, respectively.
PC-45632

Pyr10

TRPC3 inhibitor

Pyr10 is a novel TRPC3-selective inhibitor, inhibits Ca2+ influx in carbachol-stimulated TRPC3-transfected HEK293 cells with IC50 of 0.72 uM.
PC-45764

BCTC

TRPV1 antagonist

BCTC is a highly potent, selective, CNS-penetrant TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 with IC50 values of 35 and 6 nM, respectively.
PC-45355

Nonivamide

TRPV1 agonist

Nonivamide is a capsaicin analog that acts as an agonist of TRPV1 channel.
PC-25552

TRPM2 inhibitor LC4

TRPM2 inhibitor

TRPM2 inhibitor LC4 is a potent and selective TRPM2 inhibitor with IC50 of 0.66 uM, reduces the infarct volume and oxidative-stress level in transient middle cerebral artery occlusion (tMCAO) model.
PC-25551

TRPM2 inhibitor D10

TRPM2 inhibitor

TRPM2 inhibitor D10 is a highly seletive small molecule TRPM2 inhibitor with IC50 of 2.29 uM, demonstrates significant neuroprotective effects in vitro, shows robust efficacy in reducing cerebral infarction in a transient middle cerebral artery occlusion (tMCAO) model.
PC-25470

TRPA1 agonist NMTA

TRPA1 agonist

TRPA1 agonist NMTA is a selective, nonelectrophilic transient receptor potential ankyrin 1 (TRPA1) agonist with EC50 of 50.05 uM for hTRPA1, induces Ca2+ influx and exhibits antinociceptive effects.

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