Cat. No. |
Product Name |
Information |
PC-60668 |
MRS 1477
|
A small molecule positive allosteric modulator of both proton and vanilloid activation of TRPV1 (EC50=21.3 uM). |
PC-70040 |
RN-9893 hydrochloride
|
A potent, selective orally-bioavailable TRPV4 antagonist with IC50 of 320, 420 and 660 nM for mouse, human and rat TRPV4 channels, respectively. |
PC-70039 |
RN-9893
|
A potent, selective orally-bioavailable TRPV4 antagonist with IC50 of 320, 420 and 660 nM for mouse, human and rat TRPV4 channels, respectively. |
PC-45790 |
Clemizole hydrochloride
|
An H1 histamine receptor antagonist that substantially inhibits HCV replication by suppression of NS4B's RNA binding (IC50=24 nM) with little toxicity for the host cells. |
PC-45789 |
Clemizole
|
An H1 histamine receptor antagonist that substantially inhibits HCV replication by suppression of NS4B's RNA binding (IC50=24 nM) with little toxicity for the host cells. |
PC-45042 |
SN-2
|
A small molecule activator of the TRPML3 ion channel with EC50 of 1.13 uM. |
PC-42062 |
JNJ-17203212
|
A potent, selective and orally bioavailable TRPV1 receptor antagonist with IC50 of 65 nM and 102 nM for hTRPV1 and rTRPV1, respectively. |
PC-45556 |
PF-4840154
|
A potent, selective agonist of the rat (EC50=97 nM) and human (EC50=23 nM) TRPA1 channel. |
PC-42689 |
AMG 517
|
A potent and selective vanilloid receptor TRPV1 antagonist with IC50 of 0.76 nM for hTRPV1. |
PC-42931 |
SB-366791
|
A potent and selective vanilloid receptor (VR1/TRPV1) antagonist. |